An efficient and metal-free method for the direct C–N coupling of indoles with azoles to produce 2-(azol-1-yl)indoles in aqueous solution has been developed. This reaction proceeded highly regioselectively to provide a variety of indole derivatives with good to excellent yields
A facile and general method for regioselective <i>C</i>2 sulfonylation reaction of indoles mediated ...
Indoles and azaindoles undergo smooth oxidation with 2-iodoxybenzoic acid (IBX) in the presence of i...
The reaction of isatin and indoles in refluxing water/ethanol (7:3) affords 3,3'-di(indolyl)oxi...
An efficient and metal-free method for the direct C–N coupling of indoles with azoles to produce 2-(...
Azidation of indoles using iodine and copper bromide as catalysts under ambient reaction conditions ...
A metal-free one-pot oxidative cross-dehydrogenation coupling reaction for the formation of C–N/C–C ...
An efficient, atom-economic one-pot method was developed for the preparation of 7-substituted indole...
International audienceThe direct dearomative addition of arenes to the C3-position of unprotected in...
The direct introduction of alkenyl groups into theindole framework avoiding its preliminary function...
An intramolecular approach towards the regioselective construction of 2,3-diarylated indoles is r...
Copper-mediated direct and regioselective C3-cyanation of indoles using benzyl cyanide as the cyanid...
Rh(III)-catalyzed regioselective alkylation of indoles with diazo compounds as a highly efficient an...
A new protocol for the preparation of N-substituted indole-3-carboxylates has been developed. The ke...
An expeditious, functional group-tolerant synthesis of indoles from isatins is described. Isatins ar...
The aza-alkylation reaction at indole's C3 position allows the introduction of a differently substit...
A facile and general method for regioselective <i>C</i>2 sulfonylation reaction of indoles mediated ...
Indoles and azaindoles undergo smooth oxidation with 2-iodoxybenzoic acid (IBX) in the presence of i...
The reaction of isatin and indoles in refluxing water/ethanol (7:3) affords 3,3'-di(indolyl)oxi...
An efficient and metal-free method for the direct C–N coupling of indoles with azoles to produce 2-(...
Azidation of indoles using iodine and copper bromide as catalysts under ambient reaction conditions ...
A metal-free one-pot oxidative cross-dehydrogenation coupling reaction for the formation of C–N/C–C ...
An efficient, atom-economic one-pot method was developed for the preparation of 7-substituted indole...
International audienceThe direct dearomative addition of arenes to the C3-position of unprotected in...
The direct introduction of alkenyl groups into theindole framework avoiding its preliminary function...
An intramolecular approach towards the regioselective construction of 2,3-diarylated indoles is r...
Copper-mediated direct and regioselective C3-cyanation of indoles using benzyl cyanide as the cyanid...
Rh(III)-catalyzed regioselective alkylation of indoles with diazo compounds as a highly efficient an...
A new protocol for the preparation of N-substituted indole-3-carboxylates has been developed. The ke...
An expeditious, functional group-tolerant synthesis of indoles from isatins is described. Isatins ar...
The aza-alkylation reaction at indole's C3 position allows the introduction of a differently substit...
A facile and general method for regioselective <i>C</i>2 sulfonylation reaction of indoles mediated ...
Indoles and azaindoles undergo smooth oxidation with 2-iodoxybenzoic acid (IBX) in the presence of i...
The reaction of isatin and indoles in refluxing water/ethanol (7:3) affords 3,3'-di(indolyl)oxi...