A facile and general method for regioselective <i>C</i>2 sulfonylation reaction of indoles mediated by iodine is described. The 2-sulfonylated products were obtained up to 96% yield under mild reaction conditions (room temperature, 2 h)
An efficient Ir-catalyzed amidation of indoles with sulfonyl azides is disclosed, affording diverse ...
The preparation and manipulation of functionalized low molecular weight heteroaromatic compounds is ...
The Fischer indole synthesis occurs in high yield with one equivalent of the ionic liquid choline ch...
A palladium-catalyzed direct C–H bond sulfonylation of indoles with the insertion of sulfur dioxide ...
Indole derivs. I (R = H, Me; R1 = H, Me, Ph; R2 = H) were treated with DMSO and Me3SiCl to give I (s...
An efficient and metal-free method for the direct C–N coupling of indoles with azoles to produce 2-(...
Electron-rich aza-aromatic compounds such as indoles and pyrroles represent systems of particular in...
A new method for direct α-functionalization of 2,3-disubstituted indoles has been developed. The pre...
A new radical chain process catalysed by sulfonyl radicals has been used for the synthesis of functi...
This work demonstrates sulfonyl group-induced remote C(sp3)–N bond construction using a strategy of ...
An intramolecular approach towards the regioselective construction of 2,3-diarylated indoles is r...
Lodine was efficiently introduced into the methoxy substituted aromatic compounds, acetophenone, 1-i...
An efficient route to 2,3-disubstituted indoles was developed via reductive alkylation of 2-substitu...
An expeditious, functional group-tolerant synthesis of indoles from isatins is described. Isatins ar...
Halogenation of 2-trifluoromethylindole afforded 3-chloro-, 3-bromo- and 3-iodo derivatives in up to...
An efficient Ir-catalyzed amidation of indoles with sulfonyl azides is disclosed, affording diverse ...
The preparation and manipulation of functionalized low molecular weight heteroaromatic compounds is ...
The Fischer indole synthesis occurs in high yield with one equivalent of the ionic liquid choline ch...
A palladium-catalyzed direct C–H bond sulfonylation of indoles with the insertion of sulfur dioxide ...
Indole derivs. I (R = H, Me; R1 = H, Me, Ph; R2 = H) were treated with DMSO and Me3SiCl to give I (s...
An efficient and metal-free method for the direct C–N coupling of indoles with azoles to produce 2-(...
Electron-rich aza-aromatic compounds such as indoles and pyrroles represent systems of particular in...
A new method for direct α-functionalization of 2,3-disubstituted indoles has been developed. The pre...
A new radical chain process catalysed by sulfonyl radicals has been used for the synthesis of functi...
This work demonstrates sulfonyl group-induced remote C(sp3)–N bond construction using a strategy of ...
An intramolecular approach towards the regioselective construction of 2,3-diarylated indoles is r...
Lodine was efficiently introduced into the methoxy substituted aromatic compounds, acetophenone, 1-i...
An efficient route to 2,3-disubstituted indoles was developed via reductive alkylation of 2-substitu...
An expeditious, functional group-tolerant synthesis of indoles from isatins is described. Isatins ar...
Halogenation of 2-trifluoromethylindole afforded 3-chloro-, 3-bromo- and 3-iodo derivatives in up to...
An efficient Ir-catalyzed amidation of indoles with sulfonyl azides is disclosed, affording diverse ...
The preparation and manipulation of functionalized low molecular weight heteroaromatic compounds is ...
The Fischer indole synthesis occurs in high yield with one equivalent of the ionic liquid choline ch...