Additional file: of Automated synthesis of [18F]DCFPyL via direct radiofluorination and validation in preclinical prostate cancer models

Vincent Bouvet (3761455)
Melinda Wuest (1653253)
Hans-Soenke Jans (3761449)
Nancy Janzen (1428712)
Afaf Genady (3761452)
John Valliant (2355454)
Francois Benard (3761458)
Frank Wuest (1589737)

Publication date

May 2016

DOI

10.6084/m9.figshare.c.3696643_d1.v1

Abstract

Supplementary information. Automated synthesis of [18F]DCFPyL via direct radiofluorination and radiopharmacological evaluation in preclinical prostate cancer models. (DOCX 446 kb

Extracted data

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Additional file: of Automated synthesis of [18F]DCFPyL via direct radiofluorination and validation in preclinical prostate cancer models

Vincent Bouvet (3761455)
Melinda Wuest (1653253)
Hans-Soenke Jans (3761449)
Nancy Janzen (1428712)
Afaf Genady (3761452)
John Valliant (2355454)
Francois Benard (3761458)
Frank Wuest (1589737)

Open link

Publication date

May 2016

DOI

10.6084/m9.figshare.c.3696643_d1.v1

Abstract

Supplementary information. Automated synthesis of [18F]DCFPyL via direct radiofluorination and radiopharmacological evaluation in preclinical prostate cancer models. (DOCX 446 kb

Extracted data

Martina Wirtz (5556986)
Alexander Schmidt (68515)
Margret Schottelius (1816879)
Stephanie Robu (5096471)
Thomas GĂźnther (5096495)
Markus Schwaiger (10806)
Hans-JĂźrgen Wester (5096492)

August 2018

Supporting information contains the synthetic yields and exemplary illustrations of cell binding stu...

Additional file 1: of Heterogeneous drug penetrance of veliparib and carboplatin measured in triple negative breast tumors

Imke Bartelink (4428460)
Brendan Prideaux (1604743)
Gregor Krings (4428451)
Lisa Wilmes (4428430)
Pei Lee (3802915)
Pan Bo (4428466)
Byron Hann (755266)
Jean-Philippe CoppĂŠ (4428484)
Diane Heditsian (4428442)
Lamorna Swigart-Brown (732546)
Ella Jones (4428463)
Sergey Magnitsky (4428454)
Ron Keizer (4428448)
Niels de Vries (4428436)
Hilde Rosing (1519048)
Nela Pawlowska (4428445)
Scott Thomas (431824)
Mallika Dhawan (4428433)
Rahul Aggarwal (4428457)
Pamela Munster (4428439)
Laura Esserman (42231)
Weiming Ruan (2641168)
Alan Wu (526260)
Douglas Yee (312426)
VĂŠronique Dartois (3429002)
Radojka Savic (4428469)
Denise Wolf (477504)
Laura van ât Veer (4428481)

September 2017

Technical aspects of the MALDI-MSI, ICP-MS and LC-MS methods. Technical aspects of the MALDI-MSI, IC...

Additional file 1 of Boosting cisplatin chemotherapy by nanomotor-enhanced tumor penetration and DNA adducts formation

Lihua Xu (534555)
Kaixiang Zhang (1592236)
Xing Ma (540879)
Yingying Li (50341)
Yajie Jin (3628574)
Chenglin Liang (8551497)
Yong Wang (12837)
Wendi Duan (11719898)
Hongling Zhang (815356)
Zhenzhong Zhang (806974)
Jinjin Shi (815355)
Junjie Liu (193511)
Yunlong Wang (180471)
Wentao Li (1413067)

September 2022

Additional file 1: Figure S1. DLS analysis of F68@TA prepared by different mass ratio of F68 and TA....

Additional file 1: of Synthesis and preclinical evaluation of novel 18F-labeled Glu-urea-Glu-based PSMA inhibitors for prostate cancer imaging: a comparison with 18F-DCFPyl and 18F-PSMA-1007

Stephanie Robu (5096471)
Alexander Schmidt (68515)
Matthias Eiber (4896889)
Margret Schottelius (1816879)
Thomas GĂźnther (5096495)
Behrooz Hooshyar Yousefi (5096468)
Markus Schwaiger (10806)
Hans-JĂźrgen Wester (5096492)

April 2018

Supporting information contains the description of the chemical synthesis and radiolabeling of all c...

Additional file 1: of Alterations in androgen deprivation enhanced prostate-specific membrane antigen (PSMA) expression in prostate cancer cells as a target for diagnostics and therapy

B. Meller (3767254)
F. Bremmer (3767257)
C. Sahlmann (3767242)
S. Hijazi (3767245)
C. Bouter (3767263)
L. Trojan (3767251)
J. Meller (3767248)
P. Thelen (3767260)

November 2015

68 Ga-HBED-CC Radio-HPLC. Quality control of a regular Ga-HBED-CC synthesis. Radiochemical purity wa...

Automated synthesis of [18F]DCFPyL via direct radiofluorination and validation in preclinical prostate cancer models

Bouvet, Vincent
Wuest, Melinda
Jans, Hans-Soenke
Janzen, Nancy
Genady, Afaf R
Valliant, John F
Benard, Francois
Wuest, Frank

May 2016

Background: Prostate-specific membrane antigen (PSMA) is frequently overexpressed a...

Additional file 1: of Preclinical validation of 3-phosphoinositide-dependent protein kinase 1 inhibition in pancreatic cancer

Aikaterini Emmanouilidi (6701207)
Chanse Fyffe (6701210)
Riccardo Ferro (6701213)
Charlotte Edling (6701216)
Emily Capone (6701219)
Simona Sestito (1871410)
Simona Rapposelli (1577473)
Rossano Lattanzio (118191)
Stefano Iacobelli (350376)
Gianluca Sala (256062)
Tania Maffucci (104802)
Marco Falasca (104805)

May 2019

Synthetic procedure followed for the synthesis of MP7 and characterization of intermediates. (DOCX 1...

Additional file 4: of Uniform intratumoral distribution of radioactivity produced using two different radioagents, 64Cu-cyclam-RAFT-c(-RGDfK-)4 and 64Cu-ATSM, improves therapeutic efficacy in a small animal tumor model

Zhao-Hui Jin (32111)
Atsushi Tsuji (5424743)
Mélissa Degardin (5424740)
Aya Sugyo (389882)
Yukie Yoshii (416882)
Kotaro Nagatsu (399964)
Ming-Rong Zhang (136828)
Yasuhisa Fujibayashi (416891)
Pascal Dumy (8679)
Didier Boturyn (32114)
Tatsuya Higashi (5424737)

June 2018

Tumor growth curves of U87MG tumor-bearing mice after single injection of the vehicle solution (cont...

Additional file 7: of Uniform intratumoral distribution of radioactivity produced using two different radioagents, 64Cu-cyclam-RAFT-c(-RGDfK-)4 and 64Cu-ATSM, improves therapeutic efficacy in a small animal tumor model

Zhao-Hui Jin (32111)
Atsushi Tsuji (5424743)
Mélissa Degardin (5424740)
Aya Sugyo (389882)
Yukie Yoshii (416882)
Kotaro Nagatsu (399964)
Ming-Rong Zhang (136828)
Yasuhisa Fujibayashi (416891)
Pascal Dumy (8679)
Didier Boturyn (32114)
Tatsuya Higashi (5424737)

June 2018

Hematology (a) and hepatorenal functions (b) of U87MG tumor-bearing mice after co-administration of ...

Additional file 3: Table e1. of In vitro and in vivo evaluation of the radiosensitizing effect of a selective FGFR inhibitor (JNJ-42756493) for rectal cancer

Maud Verstraete (3431399)
Annelies Debucquoy (3431396)
Annelies Gonnissen (3431393)
Ruveyda Dok (3431402)
Sofie Isebaert (757211)
Ellen Devos (319514)
William McBride (486440)
Karin Haustermans (757212)

December 2015

Primer sequences, primer probes and cycling conditions used for qPCR of different genes. (DOCX 15Â k...

Additional file 1: of Initial biological evaluations of 18F-KS1, a novel ascorbate derivative to image oxidative stress in cancer

Kiran Kumar Solingapuram Sai (2411398)
Nagaraju Bashetti (6712211)
Xiaofei Chen (56655)
Skylar Norman (6712214)
Justin Hines (6712217)
Omsai Meka (6712220)
J. Kumar (1914238)
Sriram Devanathan (474812)
Gagan Deep (326431)
Cristina Furdui (159987)
Akiva Mintz (4876543)

May 2019

Figure S1. (A) Representative semiprep HPLC chromatogram with upper UV and lower radio γ trace of 18...

Additional file 2: of Synthesis and bio-molecular study of (+)-N-Acetyl-Îą-amino acid dehydroabietylamine derivative for the selective therapy of hepatocellular carcinoma

Muhammad Mustufa (3499511)
Cigdem Ozen (412802)
Imran Hashmi (765111)
Afshan Aslam (3499517)
Jameel Baig (3499514)
Gokhan Yildiz (412797)
Shoaib Muhammad (3499523)
Imam Solangi (3499526)
Naim ul Hasan Naqvi (3499520)
Mehmet Ozturk (246997)
Firdous Ali (3499529)

November 2016

Characterization and Synthesis. Spectroscopic data. Characterization of compounds through spectral d...

Additional file 1: Supplementary data on the synthesis of BODIPY-BBN, its in-vitro characterization and its in-vivo biodistribution and stability. Figure S1. of Development of a clickable bimodal fluorescent/PET probe for in vivo imaging

Andreas Paulus (3767554)
Pooja Desai (3767557)
Brandon Carney (3767551)
Giuseppe Carlucci (393306)
Thomas Reiner (1326930)
Christian Brand (1326921)
Wolfgang Weber (1390167)

August 2015

Synthesis and analytical data of BODIPY-azide 1. Figure S2. Synthesis of BODIPY-BBN 5 using CuAAC cl...

Additional file 1: of Synthesis and in vitro and in vivo evaluation of urea-based PSMA inhibitors with increased lipophilicity

Martina Wirtz (5556986)
Alexander Schmidt (68515)
Margret Schottelius (1816879)
Stephanie Robu (5096471)
Thomas GĂźnther (5096495)
Markus Schwaiger (10806)
Hans-JĂźrgen Wester (5096492)

August 2018

Supporting information contains the synthetic yields and exemplary illustrations of cell binding stu...

Additional file 1: of Heterogeneous drug penetrance of veliparib and carboplatin measured in triple negative breast tumors

Imke Bartelink (4428460)
Brendan Prideaux (1604743)
Gregor Krings (4428451)
Lisa Wilmes (4428430)
Pei Lee (3802915)
Pan Bo (4428466)
Byron Hann (755266)
Jean-Philippe CoppĂŠ (4428484)
Diane Heditsian (4428442)
Lamorna Swigart-Brown (732546)
Ella Jones (4428463)
Sergey Magnitsky (4428454)
Ron Keizer (4428448)
Niels de Vries (4428436)
Hilde Rosing (1519048)
Nela Pawlowska (4428445)
Scott Thomas (431824)
Mallika Dhawan (4428433)
Rahul Aggarwal (4428457)
Pamela Munster (4428439)
Laura Esserman (42231)
Weiming Ruan (2641168)
Alan Wu (526260)
Douglas Yee (312426)
VĂŠronique Dartois (3429002)
Radojka Savic (4428469)
Denise Wolf (477504)
Laura van ât Veer (4428481)

September 2017

Technical aspects of the MALDI-MSI, ICP-MS and LC-MS methods. Technical aspects of the MALDI-MSI, IC...

Additional file 1 of Boosting cisplatin chemotherapy by nanomotor-enhanced tumor penetration and DNA adducts formation

Lihua Xu (534555)
Kaixiang Zhang (1592236)
Xing Ma (540879)
Yingying Li (50341)
Yajie Jin (3628574)
Chenglin Liang (8551497)
Yong Wang (12837)
Wendi Duan (11719898)
Hongling Zhang (815356)
Zhenzhong Zhang (806974)
Jinjin Shi (815355)
Junjie Liu (193511)
Yunlong Wang (180471)
Wentao Li (1413067)

September 2022

Additional file 1: Figure S1. DLS analysis of F68@TA prepared by different mass ratio of F68 and TA....

Additional file 1: of Synthesis and preclinical evaluation of novel 18F-labeled Glu-urea-Glu-based PSMA inhibitors for prostate cancer imaging: a comparison with 18F-DCFPyl and 18F-PSMA-1007

Stephanie Robu (5096471)
Alexander Schmidt (68515)
Matthias Eiber (4896889)
Margret Schottelius (1816879)
Thomas GĂźnther (5096495)
Behrooz Hooshyar Yousefi (5096468)
Markus Schwaiger (10806)
Hans-JĂźrgen Wester (5096492)

April 2018

Supporting information contains the description of the chemical synthesis and radiolabeling of all c...

Additional file 1: of Alterations in androgen deprivation enhanced prostate-specific membrane antigen (PSMA) expression in prostate cancer cells as a target for diagnostics and therapy

B. Meller (3767254)
F. Bremmer (3767257)
C. Sahlmann (3767242)
S. Hijazi (3767245)
C. Bouter (3767263)
L. Trojan (3767251)
J. Meller (3767248)
P. Thelen (3767260)

November 2015

68 Ga-HBED-CC Radio-HPLC. Quality control of a regular Ga-HBED-CC synthesis. Radiochemical purity wa...

Additional file 1: of Preclinical validation of 3-phosphoinositide-dependent protein kinase 1 inhibition in pancreatic cancer

Aikaterini Emmanouilidi (6701207)
Chanse Fyffe (6701210)
Riccardo Ferro (6701213)
Charlotte Edling (6701216)
Emily Capone (6701219)
Simona Sestito (1871410)
Simona Rapposelli (1577473)
Rossano Lattanzio (118191)
Stefano Iacobelli (350376)
Gianluca Sala (256062)
Tania Maffucci (104802)
Marco Falasca (104805)

May 2019

Synthetic procedure followed for the synthesis of MP7 and characterization of intermediates. (DOCX 1...

Zhao-Hui Jin (32111)
Atsushi Tsuji (5424743)
Mélissa Degardin (5424740)
Aya Sugyo (389882)
Yukie Yoshii (416882)
Kotaro Nagatsu (399964)
Ming-Rong Zhang (136828)
Yasuhisa Fujibayashi (416891)
Pascal Dumy (8679)
Didier Boturyn (32114)
Tatsuya Higashi (5424737)

June 2018

Tumor growth curves of U87MG tumor-bearing mice after single injection of the vehicle solution (cont...

Zhao-Hui Jin (32111)
Atsushi Tsuji (5424743)
Mélissa Degardin (5424740)
Aya Sugyo (389882)
Yukie Yoshii (416882)
Kotaro Nagatsu (399964)
Ming-Rong Zhang (136828)
Yasuhisa Fujibayashi (416891)
Pascal Dumy (8679)
Didier Boturyn (32114)
Tatsuya Higashi (5424737)

June 2018

Hematology (a) and hepatorenal functions (b) of U87MG tumor-bearing mice after co-administration of ...

Additional file 3: Table e1. of In vitro and in vivo evaluation of the radiosensitizing effect of a selective FGFR inhibitor (JNJ-42756493) for rectal cancer

Maud Verstraete (3431399)
Annelies Debucquoy (3431396)
Annelies Gonnissen (3431393)
Ruveyda Dok (3431402)
Sofie Isebaert (757211)
Ellen Devos (319514)
William McBride (486440)
Karin Haustermans (757212)

December 2015

Primer sequences, primer probes and cycling conditions used for qPCR of different genes. (DOCX 15Â k...

Additional file 1: of Initial biological evaluations of 18F-KS1, a novel ascorbate derivative to image oxidative stress in cancer

Kiran Kumar Solingapuram Sai (2411398)
Nagaraju Bashetti (6712211)
Xiaofei Chen (56655)
Skylar Norman (6712214)
Justin Hines (6712217)
Omsai Meka (6712220)
J. Kumar (1914238)
Sriram Devanathan (474812)
Gagan Deep (326431)
Cristina Furdui (159987)
Akiva Mintz (4876543)

May 2019

Figure S1. (A) Representative semiprep HPLC chromatogram with upper UV and lower radio γ trace of 18...

Additional file 2: of Synthesis and bio-molecular study of (+)-N-Acetyl-Îą-amino acid dehydroabietylamine derivative for the selective therapy of hepatocellular carcinoma

Muhammad Mustufa (3499511)
Cigdem Ozen (412802)
Imran Hashmi (765111)
Afshan Aslam (3499517)
Jameel Baig (3499514)
Gokhan Yildiz (412797)
Shoaib Muhammad (3499523)
Imam Solangi (3499526)
Naim ul Hasan Naqvi (3499520)
Mehmet Ozturk (246997)
Firdous Ali (3499529)

November 2016

Characterization and Synthesis. Spectroscopic data. Characterization of compounds through spectral d...

Andreas Paulus (3767554)
Pooja Desai (3767557)
Brandon Carney (3767551)
Giuseppe Carlucci (393306)
Thomas Reiner (1326930)
Christian Brand (1326921)
Wolfgang Weber (1390167)

August 2015

Synthesis and analytical data of BODIPY-azide 1. Figure S2. Synthesis of BODIPY-BBN 5 using CuAAC cl...

Additional file 1: of Synthesis and in vitro and in vivo evaluation of urea-based PSMA inhibitors with increased lipophilicity

Martina Wirtz (5556986)
Alexander Schmidt (68515)
Margret Schottelius (1816879)
Stephanie Robu (5096471)
Thomas GĂźnther (5096495)
Markus Schwaiger (10806)
Hans-JĂźrgen Wester (5096492)

August 2018

Supporting information contains the synthetic yields and exemplary illustrations of cell binding stu...

Additional file 1: of Heterogeneous drug penetrance of veliparib and carboplatin measured in triple negative breast tumors

Imke Bartelink (4428460)
Brendan Prideaux (1604743)
Gregor Krings (4428451)
Lisa Wilmes (4428430)
Pei Lee (3802915)
Pan Bo (4428466)
Byron Hann (755266)
Jean-Philippe CoppĂŠ (4428484)
Diane Heditsian (4428442)
Lamorna Swigart-Brown (732546)
Ella Jones (4428463)
Sergey Magnitsky (4428454)
Ron Keizer (4428448)
Niels de Vries (4428436)
Hilde Rosing (1519048)
Nela Pawlowska (4428445)
Scott Thomas (431824)
Mallika Dhawan (4428433)
Rahul Aggarwal (4428457)
Pamela Munster (4428439)
Laura Esserman (42231)
Weiming Ruan (2641168)
Alan Wu (526260)
Douglas Yee (312426)
VĂŠronique Dartois (3429002)
Radojka Savic (4428469)
Denise Wolf (477504)
Laura van ât Veer (4428481)

September 2017

Technical aspects of the MALDI-MSI, ICP-MS and LC-MS methods. Technical aspects of the MALDI-MSI, IC...

Additional file 1 of Boosting cisplatin chemotherapy by nanomotor-enhanced tumor penetration and DNA adducts formation

Lihua Xu (534555)
Kaixiang Zhang (1592236)
Xing Ma (540879)
Yingying Li (50341)
Yajie Jin (3628574)
Chenglin Liang (8551497)
Yong Wang (12837)
Wendi Duan (11719898)
Hongling Zhang (815356)
Zhenzhong Zhang (806974)
Jinjin Shi (815355)
Junjie Liu (193511)
Yunlong Wang (180471)
Wentao Li (1413067)

September 2022

Additional file 1: Figure S1. DLS analysis of F68@TA prepared by different mass ratio of F68 and TA....

Additional file: of Automated synthesis of [18F]DCFPyL via direct radiofluorination and validation in preclinical prostate cancer models

Abstract

Extracted data

Additional file: of Automated synthesis of [18F]DCFPyL via direct radiofluorination and validation in preclinical prostate cancer models

Abstract

Extracted data

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