A n-BuLi triggered practical amination protocol of methoxy pyridine derivatives with aliphatic amines was developed. The reaction could finish in 30 min for primary amines and 10 min for secondary amines. The amination is further highlighted by its excellent reactivity and substrate scope.KEYWORDS: amination, methoxy pyridines, n-BuLi, transition-metal-fre
The catalytic system generated in situ from the tetranuclear Ru–H complex with a catechol ligand (1/...
(Hetero)Aryl amines, an important class of organic molecules in medicinal chemistry, are most common...
This thesis focuses on two distinct methods which were developed to access both a series of dihetero...
Among Pd-catalyzed carbon-heteroatom cross-coupling reactions, C-N bond formation, known as Buchwald...
Different substituted pyridinium N-heteroarylaminides have been prepared in one step from N-aminopyr...
The synthesis of aromatic amines is of utmost importance in a wide range of chemical contexts. We re...
A mild and highly efficient catalytic amination procedure for chloroheteroarenes at ambient temperat...
Pyridinium-N-(2´-pyridyl)aminide was reacted with different α-halocarbonyl derivatives and related c...
Buchwald–Hartwig Amination (BHA), which establishes C−N bonds between aryl halides and amines via Pd...
Tetrasubstituted N-methylpyridinium salts bearing a free tertiary amino group have been synthesized ...
The thesis is focused on hydroxylamine-mediated direct arene C-H amination and C-C amination from be...
International audiencePyridines carrying heterosubstituents (such as carboxy, amido, amino, alkoxy o...
The aliphatic amine motif is a ubiquitous and uniquely important functional group in pharmaceutical ...
The first part of this research focuses on developing efficient methods to address challenging Buchw...
A simple transition metal-free procedure using formal dehyde for the N,N-dimethylation and N-methyla...
The catalytic system generated in situ from the tetranuclear Ru–H complex with a catechol ligand (1/...
(Hetero)Aryl amines, an important class of organic molecules in medicinal chemistry, are most common...
This thesis focuses on two distinct methods which were developed to access both a series of dihetero...
Among Pd-catalyzed carbon-heteroatom cross-coupling reactions, C-N bond formation, known as Buchwald...
Different substituted pyridinium N-heteroarylaminides have been prepared in one step from N-aminopyr...
The synthesis of aromatic amines is of utmost importance in a wide range of chemical contexts. We re...
A mild and highly efficient catalytic amination procedure for chloroheteroarenes at ambient temperat...
Pyridinium-N-(2´-pyridyl)aminide was reacted with different α-halocarbonyl derivatives and related c...
Buchwald–Hartwig Amination (BHA), which establishes C−N bonds between aryl halides and amines via Pd...
Tetrasubstituted N-methylpyridinium salts bearing a free tertiary amino group have been synthesized ...
The thesis is focused on hydroxylamine-mediated direct arene C-H amination and C-C amination from be...
International audiencePyridines carrying heterosubstituents (such as carboxy, amido, amino, alkoxy o...
The aliphatic amine motif is a ubiquitous and uniquely important functional group in pharmaceutical ...
The first part of this research focuses on developing efficient methods to address challenging Buchw...
A simple transition metal-free procedure using formal dehyde for the N,N-dimethylation and N-methyla...
The catalytic system generated in situ from the tetranuclear Ru–H complex with a catechol ligand (1/...
(Hetero)Aryl amines, an important class of organic molecules in medicinal chemistry, are most common...
This thesis focuses on two distinct methods which were developed to access both a series of dihetero...
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