Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors — [34 refs. + subrefs.]. — (MILITE, C.; FEOLI, A.; VIVIANO, M.; RESCIGNO, D.; MAI, A.; CASTELLANO, S.; SBARDELLA*, G.; ChemMedChem 11 (2016) 16, 1680-1685, http://dx.doi.org/10.1002/cmdc.201600272 ; Dip. Farm., Univ. Studi Salerno, I-84084 Fisciano, Salerno, Italy; Eng.) — Koehle
Lysine Demethylases (KDMs) represent an interesting drug target as they have been implicated in many...
Epigenetic alterations relate to various human diseases, and developing inhibitors of Kme regulatory...
The development of modern pharmaceuticals relies heavily upon the drug discovery process to uncover ...
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors — [34 refs. + subrefs.]. ...
ABSTRACT: The lysine methyltransferase SETD8 is the only known methyltransfer-ase that catalyzes mon...
SETD8/SET8/Pr-SET7/KMT5A is the only known lysine methyltransferase that monomethylates lysine 20 of...
SETD8/SET8/Pr-SET7/KMT5A is the only known lysine methyltransferase that monomethylates lysine 20 of...
The lysine methyltransferase SETD8 is the only known methyltransferase that catalyzes monomethylatio...
The lysine methyltransferase SETD8 is the only known methyltransferase that catalyzes monomethylatio...
ABSTRACT: SETD8/SET8/Pr-SET7/KMT5A is the sole protein lysine methyltransferase (PKMT) known to mono...
(Chemical Equation Presented) Coding control: Protein arginine methyltransferases (PRMTs) and histon...
2015-2016 > Academic research: refereed > Publication in refereed journalVersion of RecordPublishe
*S Supporting Information ABSTRACT: Histone Nε-methyl lysine demethylases KDM2/7 have been identifie...
The epigenetic component of cancer is now well-established and epigenetic therapeutics targeting his...
The extracellular matrix (ECM) is a complex structured network of secreted macromolecules and proteo...
Lysine Demethylases (KDMs) represent an interesting drug target as they have been implicated in many...
Epigenetic alterations relate to various human diseases, and developing inhibitors of Kme regulatory...
The development of modern pharmaceuticals relies heavily upon the drug discovery process to uncover ...
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors — [34 refs. + subrefs.]. ...
ABSTRACT: The lysine methyltransferase SETD8 is the only known methyltransfer-ase that catalyzes mon...
SETD8/SET8/Pr-SET7/KMT5A is the only known lysine methyltransferase that monomethylates lysine 20 of...
SETD8/SET8/Pr-SET7/KMT5A is the only known lysine methyltransferase that monomethylates lysine 20 of...
The lysine methyltransferase SETD8 is the only known methyltransferase that catalyzes monomethylatio...
The lysine methyltransferase SETD8 is the only known methyltransferase that catalyzes monomethylatio...
ABSTRACT: SETD8/SET8/Pr-SET7/KMT5A is the sole protein lysine methyltransferase (PKMT) known to mono...
(Chemical Equation Presented) Coding control: Protein arginine methyltransferases (PRMTs) and histon...
2015-2016 > Academic research: refereed > Publication in refereed journalVersion of RecordPublishe
*S Supporting Information ABSTRACT: Histone Nε-methyl lysine demethylases KDM2/7 have been identifie...
The epigenetic component of cancer is now well-established and epigenetic therapeutics targeting his...
The extracellular matrix (ECM) is a complex structured network of secreted macromolecules and proteo...
Lysine Demethylases (KDMs) represent an interesting drug target as they have been implicated in many...
Epigenetic alterations relate to various human diseases, and developing inhibitors of Kme regulatory...
The development of modern pharmaceuticals relies heavily upon the drug discovery process to uncover ...