Add to ORKGA facile and mild synthesis of Nα-protected amino/peptide hydroxamic acids is accomplished from the corresponding Nα-protected amino/peptide thioacids using I2, 1-hydroxybenzotriazole (HOBt) and NH2OH at RT. The protocol can be extended to bifunctional as well as sterically hindered amino acids, to afford amino/peptide hydroxamic acids in good yields
Application of the Lossen rearrangement to the synthesis of N-urethane protected α-peptidyl ureas an...
The addition of N-protected amino acids to benzonitrile oxides yields activated esters, which on cou...
574-579The activation of the Nα-urethane protected (Fmoc-/Boc-/Z-/Bsmoc) α-amino acids employing 1-[...
1430-1435A facile and mild synthesis of Nα-protected amino/peptide hydroxamic acids is accomplishe...
Racemization free synthesis of Nα-protected amino hydroxamic acids from Nα-protected amino acids emp...
We report herein an efficient protocol for the synthesis of N-urethane-protected α-amino/peptide th...
One-pot preparation of N α -protected amino/peptide hydroxamic acids from corresponding carboxylic a...
Abstract: The direct conversion of simple and sterically hindered Nα-protected amino/peptide hydrox...
The direct conversion of simple and sterically hindered Nα-protected amino/peptide hydroxamic acids ...
An alternative synthesis of α,ß-unsaturated hydroxamates via cross metathesis between a class-I olef...
Thioacids derived from N-protected amino or dipeptide and tripeptide acids undergo facile N-acylatio...
Reaction of N-protected amino acids with pivalonitrile oxide affords "active esters" which are usefu...
Reaction of N-protected amino acids with pivalonitrile oxide affords "active esters" which are usefu...
The activation of the Nα-urethane protected (Fmoc-/Boc-/Z-/Bsmoc) α-amino acids employing 1-[bis(dim...
We report herein an efficient protocol for the synthesis of N-urethane-protected α-amino/peptide thi...
Application of the Lossen rearrangement to the synthesis of N-urethane protected α-peptidyl ureas an...
The addition of N-protected amino acids to benzonitrile oxides yields activated esters, which on cou...
574-579The activation of the Nα-urethane protected (Fmoc-/Boc-/Z-/Bsmoc) α-amino acids employing 1-[...
1430-1435A facile and mild synthesis of Nα-protected amino/peptide hydroxamic acids is accomplishe...
Racemization free synthesis of Nα-protected amino hydroxamic acids from Nα-protected amino acids emp...
We report herein an efficient protocol for the synthesis of N-urethane-protected α-amino/peptide th...
One-pot preparation of N α -protected amino/peptide hydroxamic acids from corresponding carboxylic a...
Abstract: The direct conversion of simple and sterically hindered Nα-protected amino/peptide hydrox...
The direct conversion of simple and sterically hindered Nα-protected amino/peptide hydroxamic acids ...
An alternative synthesis of α,ß-unsaturated hydroxamates via cross metathesis between a class-I olef...
Thioacids derived from N-protected amino or dipeptide and tripeptide acids undergo facile N-acylatio...
Reaction of N-protected amino acids with pivalonitrile oxide affords "active esters" which are usefu...
Reaction of N-protected amino acids with pivalonitrile oxide affords "active esters" which are usefu...
The activation of the Nα-urethane protected (Fmoc-/Boc-/Z-/Bsmoc) α-amino acids employing 1-[bis(dim...
We report herein an efficient protocol for the synthesis of N-urethane-protected α-amino/peptide thi...
Application of the Lossen rearrangement to the synthesis of N-urethane protected α-peptidyl ureas an...
The addition of N-protected amino acids to benzonitrile oxides yields activated esters, which on cou...
574-579The activation of the Nα-urethane protected (Fmoc-/Boc-/Z-/Bsmoc) α-amino acids employing 1-[...