5‐Oxazoyl‐sulfamates have been profiled as versatile building blocks for modifications of oxazoles with various nucleophiles. The unified approach provides a diversification platform to directly access 5‐amino‐oxazoles, 5‐oxazolyl‐sulfides, and 5‐oxazoyl‐aryl ethers from a single precursor
International audienceThe 5‐alkoxyoxazole ring system has proved to be a useful and versatile buildi...
An efficient silver mediated one-step synthesis/construction of oxazoles using α-haloketones and pri...
An efficient protocol for the synthesis of 2,5-substituted 4-acyloxazoles and the related 2,4-substi...
Reaction of methyl 2-aryl-5-(chlorosulfonyl)-1,3-oxazole-4-carboxylates with 1H-pyrazol-5-amines and...
In order to address the current downturn in the drug discovery pipeline, initiatives are being under...
The alkylation of oxazolones through an SN1 reaction by using stabilized carbocations is reported. T...
The first section describes the synthesis of the C1' to C11' side chain of leucascandrolide A. The k...
An efficient two-step palladium catalysed synthesis of 2,5-disubstituted oxazoles is reported
Synthetic methodology for the generation of novel 1,2,5-oxathiazole-S-oxides from cycloaddition of n...
In recent years, five-membered ring cyclic sulfamidate imines (5H-1,2,3-oxathiazole 2,2-dioxides) ha...
Starting from a wide range of α-acylamino amide substructures synthesized using tritylamine as an am...
The addition of various nucleophiles to a vinyl 1,2,4-oxadiazole is described. Following optimisatio...
This thesis describes the advancement of a flexible and convergent gold-catalysed synthesis of trisu...
This thesis describes investigations by the author into the preparation of the oxazole heterocyclic ...
2,4,5-Trisubstituted oxazoles were synthesized in good yields starting from alpha-methylene ketones ...
International audienceThe 5‐alkoxyoxazole ring system has proved to be a useful and versatile buildi...
An efficient silver mediated one-step synthesis/construction of oxazoles using α-haloketones and pri...
An efficient protocol for the synthesis of 2,5-substituted 4-acyloxazoles and the related 2,4-substi...
Reaction of methyl 2-aryl-5-(chlorosulfonyl)-1,3-oxazole-4-carboxylates with 1H-pyrazol-5-amines and...
In order to address the current downturn in the drug discovery pipeline, initiatives are being under...
The alkylation of oxazolones through an SN1 reaction by using stabilized carbocations is reported. T...
The first section describes the synthesis of the C1' to C11' side chain of leucascandrolide A. The k...
An efficient two-step palladium catalysed synthesis of 2,5-disubstituted oxazoles is reported
Synthetic methodology for the generation of novel 1,2,5-oxathiazole-S-oxides from cycloaddition of n...
In recent years, five-membered ring cyclic sulfamidate imines (5H-1,2,3-oxathiazole 2,2-dioxides) ha...
Starting from a wide range of α-acylamino amide substructures synthesized using tritylamine as an am...
The addition of various nucleophiles to a vinyl 1,2,4-oxadiazole is described. Following optimisatio...
This thesis describes the advancement of a flexible and convergent gold-catalysed synthesis of trisu...
This thesis describes investigations by the author into the preparation of the oxazole heterocyclic ...
2,4,5-Trisubstituted oxazoles were synthesized in good yields starting from alpha-methylene ketones ...
International audienceThe 5‐alkoxyoxazole ring system has proved to be a useful and versatile buildi...
An efficient silver mediated one-step synthesis/construction of oxazoles using α-haloketones and pri...
An efficient protocol for the synthesis of 2,5-substituted 4-acyloxazoles and the related 2,4-substi...