Synthesis and evaluation of a thio analogue of duocarmycin SA
- K. S. MacMillan
- J. P. Lajiness
- C. Lopez-Cara
- R. Romagnoli
- Wi. M. Robertson
- I. Hwang
- P. G. Baraldi
- D. L. Boger
Publication date
January 2009
DOI ISSN
0960-894X Citation count (estimate)
12Abstract
The design, synthesis, and preliminary evaluation of methyl 1,2,8,8a-tetrahydrocyclopropa[c]thieno[3,2- e]indol-4-one-6-carboxylate (CTI) derivatives are detailed representing a single atom change (N to S) embedded in the duocarmycin SA alkylation subuni
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