Add to ORKGTetra benzamidine derivatives were found to inhibit proteinase activity, cell proliferation and accumulation of the Ha-ras-1 mRNA in the FHO6T1-1 Chinese Hamster cell line, transformed with the activated human T24-Ha-ras-1 oncogene. Di- and Tri- benzamidine derivatives were also found to be potent inhibitors of proliferation of FHO6T1-1 cells. These latter compounds could be proposed as useful substrates in the synthesis of drug-conjugated monoclonal antibodies or growth factors
AbstractA series of novel amino-substituted N-aryl benzamide analogs were synthesized and evaluated ...
Two series of benzamides compounds bearing piperidine groups were synthesized and the Gli-luc lucife...
Histone deacetylase inhibitors (HDACIs) are in advanced clinical development as cancer therapeutic a...
In the present paper we have investigated the effects of aromatic tetra-amidines on attachment, ori...
We have synthesized N1-substituted benzamidines and polybenzamidines with the aim to produce antitum...
We have recently reported that aromatic polyamidines are powerful inhibitors of in vitro proliferati...
Analysis of the effects of aromatic poly-amidines exhibiting anti-proteinase activity on proliferat...
A new set of 5-(2-(pyrrolidin-1-yl)acetamido)-N-butyl-2-(substituted)benzamide and 5-(2-(piperidin-1...
Some of the biological processes which enhance the metastatic capacity of tumor cells are associated...
The cinnamoyl anthranilamides represent a class of biological active substances of great importance ...
We have previously described benzamide derivatives that in-hibited tumor necrosis factor (TNF) produ...
A series of benzamide-based histone deacetylases (HDACs) inhibitors possessing N-(aminopyridine) res...
We recently identified a polyamide-chlorambucil conjugate, 1R-Chl, which alkylates and down-regulate...
*To whom correspondence should be sent Benzidine (BZ) is a known animal and human carcinogen, and is...
AbstractInhibitors of ADP-ribosylation inhibited the myeloid differentiation of murine myelomonocyti...
AbstractA series of novel amino-substituted N-aryl benzamide analogs were synthesized and evaluated ...
Two series of benzamides compounds bearing piperidine groups were synthesized and the Gli-luc lucife...
Histone deacetylase inhibitors (HDACIs) are in advanced clinical development as cancer therapeutic a...
In the present paper we have investigated the effects of aromatic tetra-amidines on attachment, ori...
We have synthesized N1-substituted benzamidines and polybenzamidines with the aim to produce antitum...
We have recently reported that aromatic polyamidines are powerful inhibitors of in vitro proliferati...
Analysis of the effects of aromatic poly-amidines exhibiting anti-proteinase activity on proliferat...
A new set of 5-(2-(pyrrolidin-1-yl)acetamido)-N-butyl-2-(substituted)benzamide and 5-(2-(piperidin-1...
Some of the biological processes which enhance the metastatic capacity of tumor cells are associated...
The cinnamoyl anthranilamides represent a class of biological active substances of great importance ...
We have previously described benzamide derivatives that in-hibited tumor necrosis factor (TNF) produ...
A series of benzamide-based histone deacetylases (HDACs) inhibitors possessing N-(aminopyridine) res...
We recently identified a polyamide-chlorambucil conjugate, 1R-Chl, which alkylates and down-regulate...
*To whom correspondence should be sent Benzidine (BZ) is a known animal and human carcinogen, and is...
AbstractInhibitors of ADP-ribosylation inhibited the myeloid differentiation of murine myelomonocyti...
AbstractA series of novel amino-substituted N-aryl benzamide analogs were synthesized and evaluated ...
Two series of benzamides compounds bearing piperidine groups were synthesized and the Gli-luc lucife...
Histone deacetylase inhibitors (HDACIs) are in advanced clinical development as cancer therapeutic a...