Synthetic Approaches to 3‑(2-Nitroalkyl) Indoles and Their Use to Access Tryptamines and Related Bioactive Compounds

Synthesis, Reactivity and Biological Properties of Methoxy-Activated Indoles

Şengül, İbrahim Fazıl
Bingül, Murat
Kandemir, Hakan
Kumar, Naresh
Black, David StC.

January 2021

Indoles continue to play a central role in the development of new structures of chemical and biologi...

Synthesis of 3-(2-nitroalkyl) indoles by reaction of 3-(1-arylsulfonylalkyl) indoles with nitroalkanes

PALMIERI, Alessandro
PETRINI, Marino
TORREGIANI, Elisabetta

January 2007

Sulfonyl indoles act as effective precursors of vinylogous imino derivatives in the reaction with ni...

Preparation of indole-containing 3-(2-pyridyl)-1,2,4-triazines as tryptamine derivatives

Savchuk, M. I.
Kopchuk, D. S.
Krinochkin, A. P.
Kovalev, I. S.
Zyryanov, G. V.
Rusinov, V. L.
Chupakhin, O. N.
Зырянов, Г. В.

January 2019

A convenient method for obtaining new Schiff bases, comprising indole and 3-(2-pyridyl)-1,2,4-triazi...

Synthetic Approaches to 3‑(2-Nitroalkyl) Indoles and Their Use to Access Tryptamines and Related Bioactive Compounds

LANCIANESI, STEFANO
PALMIERI, Alessandro
PETRINI, Marino

January 2014

The review article presents a comprehensive survey on the preparation of 3-(2-nitroalkyl) indoles ai...

Synthesis of 7,7 '-Linked-Bis-Indoles Via 7-Tryptamines

Kandemir, Hakan
Şengül, İbrahim Fazıl
Gardner, Christopher R.
Werry, Eryn L.
Barron, Melissa L.
Kassiou, Michael
Black, David StC.

January 2016

The synthesis of 7-tryptamines was accomplished via the reduction of 7-nitrovinylindoles which were ...

Improved preparation of alkyl 2-(3-indolyl)-3-nitroalkanoates under fully heterogeneous conditions: stereoselective synthesis of alkyl (E)-2-(3-indolyl)-2-alkenoates

BALLINI, Roberto
GABRIELLI, Serena
PALMIERI, Alessandro
PETRINI, Marino

January 2008

Ethyl 3-nitro-2-alkenoates can be generated starting from nitroalkanes and ethyl 2-oxoacetate under ...

Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents

BARTOLUCCI, SILVIA
MARI, MICHELE
BEDINI, ANNALIDA
PIERSANTI, GIOVANNI
SPADONI, GILBERTO

January 2015

The selective C3-alkylation of indoles with N-protected ethanolamines involving the "borrowing hydro...

Synthesis of Tryptamine Derivatives via a Direct, One-Pot Reductive Alkylation of Indoles

Marika Righi
Francesca Topi
BARTOLUCCI, SILVIA
BEDINI, ANNALIDA
PIERSANTI, GIOVANNI
SPADONI, GILBERTO

January 2012

An efficient, one-pot reductive alkylation of indoles with N-protected aminoethyl acetals in the pre...

A Modular Approach to Highly Functionalized Indole Derivatives and Syntheses of Tryptamine-based SHIP Inhibitors

Shah, Jigisha

July 2016

Indole scaffolds are incorporated in a plethora of clinically useful natural products like ergotamin...

Pericyclic Reaction Development and Synthetic Studies Aimed at Select Tryptamine Derived Alkaloids

Kim, Simon J

March 2018

The initial section of this thesis entails pericyclic reaction development. Chapter 1 details develo...

A novel tin-mediated indole synthesis and its application to natural product synthesis

Peng, Ge

January 1996

A new indole synthesis is described. The key step involves a novel tin-mediated free radical reactio...

Organocatalytic Asymmetric Michael Addition of Aliphatic Aldehydes to Indolylnitroalkenes: Access to Contiguous Stereogenic Tryptamine Precursors

Jian Chen (15340)
Zhi-Cong Geng (1716694)
Ning Li (45258)
Xiao-Fei Huang (1980592)
Feng-Feng Pan (1980595)
Xing-Wang Wang (1538014)

March 2013

Because of the importance of the indole framework and the versatile transformation of nitro and form...

The analytical chemistry of synthetic routes to psychoactive tryptamines

Brandt, Simon D

January 2004

Many tryptamine derivatives are known to induce altered states of consciousness and the term 'halluc...

Synthesis of Chiral Tryptamines via a Regioselective Indole Alkylation

Jens Wolfard (5659514)
Jie Xu (34477)
Haiming Zhang (651820)
Cheol K. Chung (1857052)

August 2018

A practical synthesis of chiral tryptamines from simple, unprotected indoles has been developed. Ind...

Syntheses of indoles and natural indole alkaloids from 2-nitrostyrene derivatives

Rahman, S M Ashikur

January 2022

A short and flexible synthesis of 2,3-disubstituted indoles employing a Barluenga-type palladium-cat...

Synthesis, Reactivity and Biological Properties of Methoxy-Activated Indoles

Şengül, İbrahim Fazıl
Bingül, Murat
Kandemir, Hakan
Kumar, Naresh
Black, David StC.

January 2021

Indoles continue to play a central role in the development of new structures of chemical and biologi...

Synthesis of 3-(2-nitroalkyl) indoles by reaction of 3-(1-arylsulfonylalkyl) indoles with nitroalkanes

PALMIERI, Alessandro
PETRINI, Marino
TORREGIANI, Elisabetta

January 2007

Sulfonyl indoles act as effective precursors of vinylogous imino derivatives in the reaction with ni...

Preparation of indole-containing 3-(2-pyridyl)-1,2,4-triazines as tryptamine derivatives

Savchuk, M. I.
Kopchuk, D. S.
Krinochkin, A. P.
Kovalev, I. S.
Zyryanov, G. V.
Rusinov, V. L.
Chupakhin, O. N.
Зырянов, Г. В.

January 2019

A convenient method for obtaining new Schiff bases, comprising indole and 3-(2-pyridyl)-1,2,4-triazi...

Synthetic Approaches to 3‑(2-Nitroalkyl) Indoles and Their Use to Access Tryptamines and Related Bioactive Compounds

LANCIANESI, STEFANO
PALMIERI, Alessandro
PETRINI, Marino

January 2014

The review article presents a comprehensive survey on the preparation of 3-(2-nitroalkyl) indoles ai...

Synthesis of 7,7 '-Linked-Bis-Indoles Via 7-Tryptamines

Kandemir, Hakan
Şengül, İbrahim Fazıl
Gardner, Christopher R.
Werry, Eryn L.
Barron, Melissa L.
Kassiou, Michael
Black, David StC.

January 2016

The synthesis of 7-tryptamines was accomplished via the reduction of 7-nitrovinylindoles which were ...

Improved preparation of alkyl 2-(3-indolyl)-3-nitroalkanoates under fully heterogeneous conditions: stereoselective synthesis of alkyl (E)-2-(3-indolyl)-2-alkenoates

BALLINI, Roberto
GABRIELLI, Serena
PALMIERI, Alessandro
PETRINI, Marino

January 2008

Ethyl 3-nitro-2-alkenoates can be generated starting from nitroalkanes and ethyl 2-oxoacetate under ...

Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents

BARTOLUCCI, SILVIA
MARI, MICHELE
BEDINI, ANNALIDA
PIERSANTI, GIOVANNI
SPADONI, GILBERTO

January 2015

The selective C3-alkylation of indoles with N-protected ethanolamines involving the "borrowing hydro...

Synthesis of Tryptamine Derivatives via a Direct, One-Pot Reductive Alkylation of Indoles

Marika Righi
Francesca Topi
BARTOLUCCI, SILVIA
BEDINI, ANNALIDA
PIERSANTI, GIOVANNI
SPADONI, GILBERTO

January 2012

An efficient, one-pot reductive alkylation of indoles with N-protected aminoethyl acetals in the pre...

A Modular Approach to Highly Functionalized Indole Derivatives and Syntheses of Tryptamine-based SHIP Inhibitors

Shah, Jigisha

July 2016

Indole scaffolds are incorporated in a plethora of clinically useful natural products like ergotamin...

Pericyclic Reaction Development and Synthetic Studies Aimed at Select Tryptamine Derived Alkaloids

Kim, Simon J

March 2018

The initial section of this thesis entails pericyclic reaction development. Chapter 1 details develo...

A novel tin-mediated indole synthesis and its application to natural product synthesis

Peng, Ge

January 1996

A new indole synthesis is described. The key step involves a novel tin-mediated free radical reactio...

Organocatalytic Asymmetric Michael Addition of Aliphatic Aldehydes to Indolylnitroalkenes: Access to Contiguous Stereogenic Tryptamine Precursors

Jian Chen (15340)
Zhi-Cong Geng (1716694)
Ning Li (45258)
Xiao-Fei Huang (1980592)
Feng-Feng Pan (1980595)
Xing-Wang Wang (1538014)

March 2013

Because of the importance of the indole framework and the versatile transformation of nitro and form...

The analytical chemistry of synthetic routes to psychoactive tryptamines

Brandt, Simon D

January 2004

Many tryptamine derivatives are known to induce altered states of consciousness and the term 'halluc...

Synthesis of Chiral Tryptamines via a Regioselective Indole Alkylation

Jens Wolfard (5659514)
Jie Xu (34477)
Haiming Zhang (651820)
Cheol K. Chung (1857052)

August 2018

A practical synthesis of chiral tryptamines from simple, unprotected indoles has been developed. Ind...

Syntheses of indoles and natural indole alkaloids from 2-nitrostyrene derivatives

Rahman, S M Ashikur

January 2022

A short and flexible synthesis of 2,3-disubstituted indoles employing a Barluenga-type palladium-cat...

Synthesis, Reactivity and Biological Properties of Methoxy-Activated Indoles

Şengül, İbrahim Fazıl
Bingül, Murat
Kandemir, Hakan
Kumar, Naresh
Black, David StC.

January 2021

Indoles continue to play a central role in the development of new structures of chemical and biologi...

Synthesis of 3-(2-nitroalkyl) indoles by reaction of 3-(1-arylsulfonylalkyl) indoles with nitroalkanes

PALMIERI, Alessandro
PETRINI, Marino
TORREGIANI, Elisabetta

January 2007

Sulfonyl indoles act as effective precursors of vinylogous imino derivatives in the reaction with ni...

Preparation of indole-containing 3-(2-pyridyl)-1,2,4-triazines as tryptamine derivatives

Savchuk, M. I.
Kopchuk, D. S.
Krinochkin, A. P.
Kovalev, I. S.
Zyryanov, G. V.
Rusinov, V. L.
Chupakhin, O. N.
Зырянов, Г. В.

January 2019

A convenient method for obtaining new Schiff bases, comprising indole and 3-(2-pyridyl)-1,2,4-triazi...

Synthetic Approaches to 3‑(2-Nitroalkyl) Indoles and Their Use to Access Tryptamines and Related Bioactive Compounds

Abstract

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Synthetic Approaches to 3‑(2-Nitroalkyl) Indoles and Their Use to Access Tryptamines and Related Bioactive Compounds

Abstract

Extracted data

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