A copper(I)-mediated one-pot synthesis of 2,3-dihydro-1H-indazole heterocycles has been developed. This synthetic route provides the desired indazoles in moderate to good yields (55%–72%) which are substantially better than those achievable with an alternative two-step reaction sequence. The reaction is tolerant of functionality on the aromatic ring
E f f i c i e n t S y n t h e s i s o f 7-S u b s t i t u t e d o r 3 , 7-D i s u b s t i t u t e d ...
We described two orthogonal heterocycle syntheses, where an arene bearing both an alkyne and a triaz...
E f f i c i e n t S y n t h e s i s o f 7-S u b s t i t u t e d o r 3 , 7-D i s u b s t i t u t e d ...
International audienceA set of variously substituted indazoles and hetero-aromatic derivatives were ...
An efficient route to substituted 1-aryl-1H-indazoles has been developed and optimized. The method i...
An efficient route to substituted 1-aryl-1H-indazoles has been developed and optimized. The method i...
We have described a facile, microwave-assisted, catalyst-free and solvent-free approach to 2H-indazo...
A one-pot–three-step method has been developed for the conversion of oxazolino-2<i>H</i>-indazoles i...
A novel and efficient method for the one-pot synthesis of 2<i>H</i>-indazole from readily available ...
A simple and efficient synthesis of 2H-indazoles is achieved from 2-primary amines, bromobenzaldehyd...
A novel and efficient method for the one-pot synthesis of 2<i>H</i>-indazole from readily available ...
Nitrosobenzenes have been used as a convenient aminating reagent for the efficient synthesis of 1H-i...
A novel and efficient method for the one-pot synthesis of 2<i>H</i>-indazole from readily available ...
A novel and efficient method for the one-pot synthesis of 2<i>H</i>-indazole from readily available ...
A simple and efficient synthesis of 2H-indazoles is achieved from 2-primary amines, bromobenzaldehyd...
E f f i c i e n t S y n t h e s i s o f 7-S u b s t i t u t e d o r 3 , 7-D i s u b s t i t u t e d ...
We described two orthogonal heterocycle syntheses, where an arene bearing both an alkyne and a triaz...
E f f i c i e n t S y n t h e s i s o f 7-S u b s t i t u t e d o r 3 , 7-D i s u b s t i t u t e d ...
International audienceA set of variously substituted indazoles and hetero-aromatic derivatives were ...
An efficient route to substituted 1-aryl-1H-indazoles has been developed and optimized. The method i...
An efficient route to substituted 1-aryl-1H-indazoles has been developed and optimized. The method i...
We have described a facile, microwave-assisted, catalyst-free and solvent-free approach to 2H-indazo...
A one-pot–three-step method has been developed for the conversion of oxazolino-2<i>H</i>-indazoles i...
A novel and efficient method for the one-pot synthesis of 2<i>H</i>-indazole from readily available ...
A simple and efficient synthesis of 2H-indazoles is achieved from 2-primary amines, bromobenzaldehyd...
A novel and efficient method for the one-pot synthesis of 2<i>H</i>-indazole from readily available ...
Nitrosobenzenes have been used as a convenient aminating reagent for the efficient synthesis of 1H-i...
A novel and efficient method for the one-pot synthesis of 2<i>H</i>-indazole from readily available ...
A novel and efficient method for the one-pot synthesis of 2<i>H</i>-indazole from readily available ...
A simple and efficient synthesis of 2H-indazoles is achieved from 2-primary amines, bromobenzaldehyd...
E f f i c i e n t S y n t h e s i s o f 7-S u b s t i t u t e d o r 3 , 7-D i s u b s t i t u t e d ...
We described two orthogonal heterocycle syntheses, where an arene bearing both an alkyne and a triaz...
E f f i c i e n t S y n t h e s i s o f 7-S u b s t i t u t e d o r 3 , 7-D i s u b s t i t u t e d ...
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