Synthesis and in vitro antimycobacterial activity of novel 3-(1H-pyrrol-1-yl)-2-oxazolidinone analogues of PNU-100480

Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones

CASTAGNOLO D
BECHI B
PAGANO M
DE LOGU A
MELEDDU R
SADDI M
BOTTA M.
MANETTI, FABRIZIO
BOTTA, MAURIZIO

January 2009

Two series of novel rigid pyrazolone derivatives were synthesized and evaluated as inhibitors of Myc...

Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: part 2. Synthesis of rigid pyrazolones

Castagnolo D
Manetti F
Radi M
Bechi B
Pagano M
Saddi M
Botta M.
DE LOGU, ALESSANDRO
MELEDDU, RITA

January 2009

Two series of novel rigid pyrazolone derivatives were synthesized and evaluated as inhibitors of Myc...

Pyrrole compounds as inhibitors of mycobacteria, synthesis thereof ans intermediates thereto

Biava M
Porretta GC
Pompei R
De Logu A.
BOTTA, MAURIZIO
MANETTI, FABRIZIO

January 2013

The present invention concerns novel pyrrole compounds, derivatives of 1-{[1,5-bis(4-chlorophenyl)-2...

Synthesis and in vitro antimycobacterial activity of novel 3-(1H-pyrrol-1-yl)-2-oxazolidinone analogues of PNU-100480

Sbardella, Gianluca
Mai, Antonello
Artico, Marino
Loddo, Roberta
Setzu, Maria Giovanna
La Colla, Paolo

January 2004

Pursuing our search program for new antitubercular drugs we decided to explore the potentiality of o...

Synthesis and in vitro evaluation of the antitubercular and antibacterial activity of novel oxazolidinones bearing octahydrocyclopenta[c]pyrrol-2-yl moieties.

조상래

January 2014

A novel series of oxazolidinone-class antimicrobial agents with 5-substituted octahydrocyclopenta[c]...

Synthesis and in vitro antibacterial activity of novel 3-azabicyclo[3.3.0]octanyl oxazolidinones.

오태권
조상래

January 2012

We synthesized a series of oxazolidinone-type antibacterials in which morpholine C-ring of linezolid...

Anti-tubercular agents. Part 6: Synthesis and antimycobacterial activity of novel arylsulfonamido conjugated oxazolidinones

Kamal, Ahmed
Shetti, Rajesh V.C.R.N.C.
Azeeza, Shaik
Swapna, P.
Khan, M. Naseer A.
Khan, Inshad Ali
Sharma, Sandeep
Abdullah, Sheikh Tasduq

January 2011

As a part of investigation of new anti-tubercular agents in this laboratory, herein we describe the ...

Antimycobacterial Agents. Novel Diarylpyrrole Derivatives of BM212 Endowed with High Activity toward Mycobacterium tuberculosis and Low Cytotoxicity

Biava, M.
Porretta, G. C.
Poce, G.
Supino, S.
Deidda, D.
Pompei, R.
Molicotti, P.
Manetti, Fabrizio
Botta, Maurizio

January 2006

On the basis of suggestions derived either from a pharmacophoric model for antitubercular agents or ...

New derivatives of BM212. a class of antimycobacterial compounds based on the pyrrole ring as a scaffold

Biava, M
PORRETTA G., C
Manetti, Fabrizio

January 2007

During our investigation in the area of antimycobacterial agents, we have identified the 1,5-(4-chlo...

Synthesis and Antibacterial Activity of Novel 2-Oxo-pyrrolidinyl Oxazolidinones

오태권
조상래

January 2012

Novel antibacterial oxazolidinones bearing pyrrolidinone ring system at the C-5 side chain were synt...

Synthesis and molecular modeling studies of novel pyrrole analogs as antimycobacterial agents

Joshi, Shrinivas D.
More, Uttam A.
Pansuriya, Ketan
Aminabhavi, Tejraj M.
Gadad, Andanappa K.

January 2017

AbstractIn the present investigation, a series of 4-(4-pyrrol-1-yl/2,5-dimethyl-4-pyrrol-1-yl) benzo...

Antimycobacterial Activities of Novel 5-(1H-1,2,3-Triazolyl)Methyl Oxazolidinones

Oludotun Adebayo Phillips
Edet Ekpenyong Udo
Reny Varghese

April 2020

The antibacterial activities of a series of triazolyl oxazolidinones against Mycobacterium tuberculo...

Synthesis and evaluation of some novel substituted 1,3,4-oxadiazole and pyrazole derivatives for antitubercular activity

Pattan, Shashikant R
Rabara, P A
Pattan, Jayashri S
Bukitagar, A A
Wakale, V S
Musmade, D S

October 2009

1453-1456A series of 1,3,4-oxadiazole and pyrazole derivatives have been synthesized and evaluated f...

Synthesis and in vitro antimycobacterial activity of some pyridine and pyrazinecarboxylic acid isosteres

Gezginci, Mikail Hakan
Gezginci, Mikail Hakan

January 1999

Tuberculosis has been one of the most commonly encountered infectious diseases of humans throughout ...

In Vitro and In Vivo Activities of Three Oxazolidinones against

Nonreplicating Mycobacterium Tuberculosis
V. Balasubramanian
B Stewart T. Colea

September 2016

Oxazolidinones represent a new class of antituberculosis drugs that exert their function by inhibiti...

Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones

CASTAGNOLO D
BECHI B
PAGANO M
DE LOGU A
MELEDDU R
SADDI M
BOTTA M.
MANETTI, FABRIZIO
BOTTA, MAURIZIO

January 2009

Two series of novel rigid pyrazolone derivatives were synthesized and evaluated as inhibitors of Myc...

Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: part 2. Synthesis of rigid pyrazolones

Castagnolo D
Manetti F
Radi M
Bechi B
Pagano M
Saddi M
Botta M.
DE LOGU, ALESSANDRO
MELEDDU, RITA

January 2009

Two series of novel rigid pyrazolone derivatives were synthesized and evaluated as inhibitors of Myc...

Pyrrole compounds as inhibitors of mycobacteria, synthesis thereof ans intermediates thereto

Biava M
Porretta GC
Pompei R
De Logu A.
BOTTA, MAURIZIO
MANETTI, FABRIZIO

January 2013

The present invention concerns novel pyrrole compounds, derivatives of 1-{[1,5-bis(4-chlorophenyl)-2...

Synthesis and in vitro antimycobacterial activity of novel 3-(1H-pyrrol-1-yl)-2-oxazolidinone analogues of PNU-100480

Sbardella, Gianluca
Mai, Antonello
Artico, Marino
Loddo, Roberta
Setzu, Maria Giovanna
La Colla, Paolo

January 2004

Pursuing our search program for new antitubercular drugs we decided to explore the potentiality of o...

Synthesis and in vitro evaluation of the antitubercular and antibacterial activity of novel oxazolidinones bearing octahydrocyclopenta[c]pyrrol-2-yl moieties.

조상래

January 2014

A novel series of oxazolidinone-class antimicrobial agents with 5-substituted octahydrocyclopenta[c]...

Synthesis and in vitro antibacterial activity of novel 3-azabicyclo[3.3.0]octanyl oxazolidinones.

오태권
조상래

January 2012

We synthesized a series of oxazolidinone-type antibacterials in which morpholine C-ring of linezolid...

Anti-tubercular agents. Part 6: Synthesis and antimycobacterial activity of novel arylsulfonamido conjugated oxazolidinones

Kamal, Ahmed
Shetti, Rajesh V.C.R.N.C.
Azeeza, Shaik
Swapna, P.
Khan, M. Naseer A.
Khan, Inshad Ali
Sharma, Sandeep
Abdullah, Sheikh Tasduq

January 2011

As a part of investigation of new anti-tubercular agents in this laboratory, herein we describe the ...

Antimycobacterial Agents. Novel Diarylpyrrole Derivatives of BM212 Endowed with High Activity toward Mycobacterium tuberculosis and Low Cytotoxicity

Biava, M.
Porretta, G. C.
Poce, G.
Supino, S.
Deidda, D.
Pompei, R.
Molicotti, P.
Manetti, Fabrizio
Botta, Maurizio

January 2006

On the basis of suggestions derived either from a pharmacophoric model for antitubercular agents or ...

New derivatives of BM212. a class of antimycobacterial compounds based on the pyrrole ring as a scaffold

Biava, M
PORRETTA G., C
Manetti, Fabrizio

January 2007

During our investigation in the area of antimycobacterial agents, we have identified the 1,5-(4-chlo...

Synthesis and Antibacterial Activity of Novel 2-Oxo-pyrrolidinyl Oxazolidinones

오태권
조상래

January 2012

Novel antibacterial oxazolidinones bearing pyrrolidinone ring system at the C-5 side chain were synt...

Synthesis and molecular modeling studies of novel pyrrole analogs as antimycobacterial agents

Joshi, Shrinivas D.
More, Uttam A.
Pansuriya, Ketan
Aminabhavi, Tejraj M.
Gadad, Andanappa K.

January 2017

AbstractIn the present investigation, a series of 4-(4-pyrrol-1-yl/2,5-dimethyl-4-pyrrol-1-yl) benzo...

Antimycobacterial Activities of Novel 5-(1H-1,2,3-Triazolyl)Methyl Oxazolidinones

Oludotun Adebayo Phillips
Edet Ekpenyong Udo
Reny Varghese

April 2020

The antibacterial activities of a series of triazolyl oxazolidinones against Mycobacterium tuberculo...

Synthesis and evaluation of some novel substituted 1,3,4-oxadiazole and pyrazole derivatives for antitubercular activity

Pattan, Shashikant R
Rabara, P A
Pattan, Jayashri S
Bukitagar, A A
Wakale, V S
Musmade, D S

October 2009

1453-1456A series of 1,3,4-oxadiazole and pyrazole derivatives have been synthesized and evaluated f...

Synthesis and in vitro antimycobacterial activity of some pyridine and pyrazinecarboxylic acid isosteres

Gezginci, Mikail Hakan
Gezginci, Mikail Hakan

January 1999

Tuberculosis has been one of the most commonly encountered infectious diseases of humans throughout ...

In Vitro and In Vivo Activities of Three Oxazolidinones against

Nonreplicating Mycobacterium Tuberculosis
V. Balasubramanian
B Stewart T. Colea

September 2016

Oxazolidinones represent a new class of antituberculosis drugs that exert their function by inhibiti...

Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones

CASTAGNOLO D
BECHI B
PAGANO M
DE LOGU A
MELEDDU R
SADDI M
BOTTA M.
MANETTI, FABRIZIO
BOTTA, MAURIZIO

January 2009

Two series of novel rigid pyrazolone derivatives were synthesized and evaluated as inhibitors of Myc...

Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: part 2. Synthesis of rigid pyrazolones

Castagnolo D
Manetti F
Radi M
Bechi B
Pagano M
Saddi M
Botta M.
DE LOGU, ALESSANDRO
MELEDDU, RITA

January 2009

Two series of novel rigid pyrazolone derivatives were synthesized and evaluated as inhibitors of Myc...

Pyrrole compounds as inhibitors of mycobacteria, synthesis thereof ans intermediates thereto

Biava M
Porretta GC
Pompei R
De Logu A.
BOTTA, MAURIZIO
MANETTI, FABRIZIO

January 2013

The present invention concerns novel pyrrole compounds, derivatives of 1-{[1,5-bis(4-chlorophenyl)-2...

Synthesis and in vitro antimycobacterial activity of novel 3-(1H-pyrrol-1-yl)-2-oxazolidinone analogues of PNU-100480

Abstract

Extracted data

Synthesis and in vitro antimycobacterial activity of novel 3-(1H-pyrrol-1-yl)-2-oxazolidinone analogues of PNU-100480

Abstract

Extracted data

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