Both enantiomers of the heterocyclic GABA analogue homo-b-proline (3-pyrrolidineacetic acid) were synthesized by a chemoenzymatic method involving the use of two enantiocomplementary enzymes in the disymmetric hydrolyses of 3-nitromethylglutaric acid diethyl este
Esterase from Horse Liver (HLAP) was able to hydrolyze a series of linear and cyclic b,b-dialkyl-c-n...
Weiss M, Gröger H. Practical, Highly Enantioselective Chemoenzymatic One-Pot Synthesis of Short-Chai...
International audienceScalable synthesis of enantiopure ( R ) and ( S )-α-Tfm-proline and α-Tfm-pipe...
Both enantiomers of the pharmacologically active GABA analogues 4-amino-3-phenyl and 4-amino-3-(4-ch...
Both enantiomerically pure antipodes of GABA analogues were prepared as hydrochloride salts, by enzy...
An enantioselective three-step synthesis of the GABA uptake inhibitor (S)-(+)-homo-beta-proline was ...
An enantioselective three-step synthesis of the GABA uptake inhibitor (<i>S</i>)-(+)-homo-β-proline ...
Chiral γ-aminobutyric acid (GABA) analogues represent abundantly prescribed drugs, which are broadly...
Chiral γ-aminobutyric acid (GABA) analogues represent abundantly prescribed drugs, which are broadly...
Starting from easily available ethyl 2-methyl-4,4,4-trifluoroacetoacetate and benzylamine each of th...
The synthesis of both enantiomers of N-benzyl-3-hydroxypyrrolidine and N-benzyl-3-hydroxypiperidine ...
Chiral γ-aminobutyric acid (GABA) analogues represent abundantly prescribed drugs, which are broadly...
Enantiopure (99% ee) cis- and trans-gamma-benzylparaconic acids and their ethyl esters were synthesi...
Enantioselective Synthesis of Endo-Cyclic Beta-Amino Acids with Two Contiguous Stereocenters via Hyd...
Enantiomerically pure L- and D-4-fluoro-3-nitrophenylalanines and L- and D-3-fluoro-4-nitrophenylala...
Esterase from Horse Liver (HLAP) was able to hydrolyze a series of linear and cyclic b,b-dialkyl-c-n...
Weiss M, Gröger H. Practical, Highly Enantioselective Chemoenzymatic One-Pot Synthesis of Short-Chai...
International audienceScalable synthesis of enantiopure ( R ) and ( S )-α-Tfm-proline and α-Tfm-pipe...
Both enantiomers of the pharmacologically active GABA analogues 4-amino-3-phenyl and 4-amino-3-(4-ch...
Both enantiomerically pure antipodes of GABA analogues were prepared as hydrochloride salts, by enzy...
An enantioselective three-step synthesis of the GABA uptake inhibitor (S)-(+)-homo-beta-proline was ...
An enantioselective three-step synthesis of the GABA uptake inhibitor (<i>S</i>)-(+)-homo-β-proline ...
Chiral γ-aminobutyric acid (GABA) analogues represent abundantly prescribed drugs, which are broadly...
Chiral γ-aminobutyric acid (GABA) analogues represent abundantly prescribed drugs, which are broadly...
Starting from easily available ethyl 2-methyl-4,4,4-trifluoroacetoacetate and benzylamine each of th...
The synthesis of both enantiomers of N-benzyl-3-hydroxypyrrolidine and N-benzyl-3-hydroxypiperidine ...
Chiral γ-aminobutyric acid (GABA) analogues represent abundantly prescribed drugs, which are broadly...
Enantiopure (99% ee) cis- and trans-gamma-benzylparaconic acids and their ethyl esters were synthesi...
Enantioselective Synthesis of Endo-Cyclic Beta-Amino Acids with Two Contiguous Stereocenters via Hyd...
Enantiomerically pure L- and D-4-fluoro-3-nitrophenylalanines and L- and D-3-fluoro-4-nitrophenylala...
Esterase from Horse Liver (HLAP) was able to hydrolyze a series of linear and cyclic b,b-dialkyl-c-n...
Weiss M, Gröger H. Practical, Highly Enantioselective Chemoenzymatic One-Pot Synthesis of Short-Chai...
International audienceScalable synthesis of enantiopure ( R ) and ( S )-α-Tfm-proline and α-Tfm-pipe...
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