Synthesis of 2-monosubstituted indolin-3-ones by cine-substitution of 3-azido-2-methoxyindolines

Yamashiro, Toshiki
Abe, Takumi
Sawada, Daisuke

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Publication date

January 2022

DOI

10.1039/d2qo00048b

Publisher

Royal Society of Chemistry (RSC)

Journal

Organic Chemistry Frontiers

Abstract

We report herein a formal cine-substitution/hydrolysis of 3-azidoindoles generated from 3-azido-2-methoxyindolines (AZINs). This protocol enables the introduction of various carboxylic acids and alcohols into indolin-3-ones at the C2-position, affording 2-monoacyloxy or alkoxy indolin-3-ones

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Synthesis of 2-monosubstituted indolin-3-ones by cine-substitution of 3-azido-2-methoxyindolines

Abstract

Extracted data

Synthesis of 2-monosubstituted indolin-3-ones by cine-substitution of 3-azido-2-methoxyindolines

Abstract

Extracted data

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