Add to ORKGA n-BuLi triggered practical amination protocol of methoxy pyridine derivatives with aliphatic amines was developed. The reaction could finish in 30 min for primary amines and 10 min for secondary amines. The amination is further highlighted by its excellent reactivity and substrate scope.KEYWORDS: amination, methoxy pyridines, n-BuLi, transition-metal-fre
Pyridinium-N-(2´-pyridyl)aminide was reacted with different α-halocarbonyl derivatives and related c...
The thesis is focused on hydroxylamine-mediated direct arene C-H amination and C-C amination from be...
International audiencePyridines carrying heterosubstituents (such as carboxy, amido, amino, alkoxy o...
Among Pd-catalyzed carbon-heteroatom cross-coupling reactions, C-N bond formation, known as Buchwald...
Different substituted pyridinium N-heteroarylaminides have been prepared in one step from N-aminopyr...
Different substituted pyridinium N-heteroarylaminides have been prepared in one step from N-aminopyr...
Different substituted pyridinium N-heteroarylaminides have been prepared in one step from N-aminopyr...
Different substituted pyridinium N-heteroarylaminides have been prepared in one step from N-aminopyr...
The synthesis of aromatic amines is of utmost importance in a wide range of chemical contexts. We re...
A mild and highly efficient catalytic amination procedure for chloroheteroarenes at ambient temperat...
Pyridinium-N-(2´-pyridyl)aminide was reacted with different α-halocarbonyl derivatives and related c...
Pyridinium-N-(2´-pyridyl)aminide was reacted with different α-halocarbonyl derivatives and related c...
Buchwald–Hartwig Amination (BHA), which establishes C−N bonds between aryl halides and amines via Pd...
Tetrasubstituted N-methylpyridinium salts bearing a free tertiary amino group have been synthesized ...
Pyridinium-N-(2´-pyridyl)aminide was reacted with different α-halocarbonyl derivatives and related c...
Pyridinium-N-(2´-pyridyl)aminide was reacted with different α-halocarbonyl derivatives and related c...
The thesis is focused on hydroxylamine-mediated direct arene C-H amination and C-C amination from be...
International audiencePyridines carrying heterosubstituents (such as carboxy, amido, amino, alkoxy o...
Among Pd-catalyzed carbon-heteroatom cross-coupling reactions, C-N bond formation, known as Buchwald...
Different substituted pyridinium N-heteroarylaminides have been prepared in one step from N-aminopyr...
Different substituted pyridinium N-heteroarylaminides have been prepared in one step from N-aminopyr...
Different substituted pyridinium N-heteroarylaminides have been prepared in one step from N-aminopyr...
Different substituted pyridinium N-heteroarylaminides have been prepared in one step from N-aminopyr...
The synthesis of aromatic amines is of utmost importance in a wide range of chemical contexts. We re...
A mild and highly efficient catalytic amination procedure for chloroheteroarenes at ambient temperat...
Pyridinium-N-(2´-pyridyl)aminide was reacted with different α-halocarbonyl derivatives and related c...
Pyridinium-N-(2´-pyridyl)aminide was reacted with different α-halocarbonyl derivatives and related c...
Buchwald–Hartwig Amination (BHA), which establishes C−N bonds between aryl halides and amines via Pd...
Tetrasubstituted N-methylpyridinium salts bearing a free tertiary amino group have been synthesized ...
Pyridinium-N-(2´-pyridyl)aminide was reacted with different α-halocarbonyl derivatives and related c...
Pyridinium-N-(2´-pyridyl)aminide was reacted with different α-halocarbonyl derivatives and related c...
The thesis is focused on hydroxylamine-mediated direct arene C-H amination and C-C amination from be...
International audiencePyridines carrying heterosubstituents (such as carboxy, amido, amino, alkoxy o...