The amino azanoradamantane hexahydro-2,5b-methano-IH-3aS,3aa,6aa-cyclopenta-[clpyrrole-4a-amine 1and the corresponding enantiomer ent-1 have been prepared along with benzamide derivatives SC-52491and SC-52490, respectively, which are of pharmaceutical interest. The key meso-azabicyclo[3.3.0] intermediate 3 was prepared via three separate routes: a [3+2] cycloaddition route, a radical cyclization/ionic cyclization route, and a reductive Pauson-Khand route
The enantioselective synthesis of advanced tetracyclic precursors of madangamine D, bearing rings AB...
A multicomponent 1,3-dipolar cycloaddition between heterocyclic aldehydes, amino esters and dipolaro...
The first half of this product was conducted at the University of East Anglia under the supervision ...
A racemic synthesis of azanoradamantane (±)-3 was accomplished via Yamamoto\u27s MAD-catalyzed Diels...
An enantioselective formal synthesis of the marine alkaloid madangamine A using phenylglycinol-deriv...
International audienceWe report the first enantioselective organocatalyzed domino synthesis of azepa...
A concise route toward two advanced fragments in the context of the total synthesis of the unique na...
textA novel application of the Pauson-Khand reaction was applied to the synthesis of a series of bri...
The 1,3-dipolar cycloaddition reaction of Substituted benzyl azides and quomarinee was studied . W...
2-Substituted azetidin-3-ones can be prepared in good yields and enantioselectivities (up to 85% ee)...
Functionalized piperidines, azepanes, azamacrocycles, morpholines, and thiomorpholines are common st...
The dissertation describes asymmetric synthesis towards C29-C34 moiety of fragment A of the Antascom...
The synthesis of enantiopure ABCE and ABCD tetracyclic advanced intermediates en route to madangamin...
I. Asymmetric Synthesis of the Aminocyclitol Pactamycin, a Universal Translocation Inhibitor A conci...
L'objectif de cette thèse de doctorat a été la mise au point de nouvelles méthodologies de synthèse ...
The enantioselective synthesis of advanced tetracyclic precursors of madangamine D, bearing rings AB...
A multicomponent 1,3-dipolar cycloaddition between heterocyclic aldehydes, amino esters and dipolaro...
The first half of this product was conducted at the University of East Anglia under the supervision ...
A racemic synthesis of azanoradamantane (±)-3 was accomplished via Yamamoto\u27s MAD-catalyzed Diels...
An enantioselective formal synthesis of the marine alkaloid madangamine A using phenylglycinol-deriv...
International audienceWe report the first enantioselective organocatalyzed domino synthesis of azepa...
A concise route toward two advanced fragments in the context of the total synthesis of the unique na...
textA novel application of the Pauson-Khand reaction was applied to the synthesis of a series of bri...
The 1,3-dipolar cycloaddition reaction of Substituted benzyl azides and quomarinee was studied . W...
2-Substituted azetidin-3-ones can be prepared in good yields and enantioselectivities (up to 85% ee)...
Functionalized piperidines, azepanes, azamacrocycles, morpholines, and thiomorpholines are common st...
The dissertation describes asymmetric synthesis towards C29-C34 moiety of fragment A of the Antascom...
The synthesis of enantiopure ABCE and ABCD tetracyclic advanced intermediates en route to madangamin...
I. Asymmetric Synthesis of the Aminocyclitol Pactamycin, a Universal Translocation Inhibitor A conci...
L'objectif de cette thèse de doctorat a été la mise au point de nouvelles méthodologies de synthèse ...
The enantioselective synthesis of advanced tetracyclic precursors of madangamine D, bearing rings AB...
A multicomponent 1,3-dipolar cycloaddition between heterocyclic aldehydes, amino esters and dipolaro...
The first half of this product was conducted at the University of East Anglia under the supervision ...