N-substituted pyrroles prepared from α-amino acids are converted to their mixed anhydrides by treatment with an acid chloride and base. Subsequent treatment with AlCl3 brings about rearrangement to the corresponding 2-acyl derivatives in overall yields of 55-81%
A variety of 3-aryl-3-chloropropeniminium salts react with α-amino acid esters under basic condition...
An efficient synthesis of 2,2'-dipyrryl ketones has been carried out from pyrrole-2-carboxylic ...
Both pyrophosphoryl chloride and phosphorus oxychloride react with aryl aliphatic acids to form mixe...
Pyrrole and its derivatives react smoothly with acid chlorides and sulfonyl chlorides in the presenc...
2-Ethanolamine and (2R)-2-aminopropanol were converted into their N-pyrrole derivatives, 14 and 15, ...
The conversion of the amino group of chiral amines, amino alcohols, amino acids and their esters int...
A variety of 2-substituted vinamidinium salts react with a-amino acid esters under basic conditions ...
Pyrrole, pyrrolidine, and indolizidine alkaloids represent important classes of natural products. Hi...
International audienceA diversity of new functionalized acyclic chiral pyrroloamide compounds were s...
Functionalization of pyrroles introducing a 2-nitroalkyl moiety allows the formation of nitro-contai...
The partial reduction of N-Boc pyrroles has been explored giving stereoselective routes to disubstit...
In the past few decades, an extensive family of structurally intriguing and biologically active pyrr...
The acylketene S,N-acetals 1a-c react with maleic anhydride (2) in refluxing acetonitrile to give th...
Acylation of O,N-acetal 1 gives excellent yields of the C-7 substituted products 2a,b. Alkylation of...
Herein, we present a new general and efficient protocol to synthesize pyrrole-2-acetic acid derivati...
A variety of 3-aryl-3-chloropropeniminium salts react with α-amino acid esters under basic condition...
An efficient synthesis of 2,2'-dipyrryl ketones has been carried out from pyrrole-2-carboxylic ...
Both pyrophosphoryl chloride and phosphorus oxychloride react with aryl aliphatic acids to form mixe...
Pyrrole and its derivatives react smoothly with acid chlorides and sulfonyl chlorides in the presenc...
2-Ethanolamine and (2R)-2-aminopropanol were converted into their N-pyrrole derivatives, 14 and 15, ...
The conversion of the amino group of chiral amines, amino alcohols, amino acids and their esters int...
A variety of 2-substituted vinamidinium salts react with a-amino acid esters under basic conditions ...
Pyrrole, pyrrolidine, and indolizidine alkaloids represent important classes of natural products. Hi...
International audienceA diversity of new functionalized acyclic chiral pyrroloamide compounds were s...
Functionalization of pyrroles introducing a 2-nitroalkyl moiety allows the formation of nitro-contai...
The partial reduction of N-Boc pyrroles has been explored giving stereoselective routes to disubstit...
In the past few decades, an extensive family of structurally intriguing and biologically active pyrr...
The acylketene S,N-acetals 1a-c react with maleic anhydride (2) in refluxing acetonitrile to give th...
Acylation of O,N-acetal 1 gives excellent yields of the C-7 substituted products 2a,b. Alkylation of...
Herein, we present a new general and efficient protocol to synthesize pyrrole-2-acetic acid derivati...
A variety of 3-aryl-3-chloropropeniminium salts react with α-amino acid esters under basic condition...
An efficient synthesis of 2,2'-dipyrryl ketones has been carried out from pyrrole-2-carboxylic ...
Both pyrophosphoryl chloride and phosphorus oxychloride react with aryl aliphatic acids to form mixe...