Add to ORKG[Abstract] Functionalization of 7-azaindole utilizing Reissert-Henze type reaction was studied. It was found that the direct halogenation, cyanation, and thiocyanation of 7-azaindole proceeded regioselectively. In chlorination of 7-azaindole, the regioselectivity was controlled by chlorination reagents as well as acylation reagents. These functional groups could be chemically modified to useful substituents
Herein we report a novel iridium(III)-catalyzed ortho-mono-alkynylation of 7-azaindoles under mild c...
A series of 3-(2-haloalkenyl)-2-pyridyl-halides undergo consecutive palladium-catalysed inter- and i...
The functionalization of arenes and heterocycles via direct C-H activation is a valuable tool in med...
An efficient and practical route to 7-azaindole framework has been developed by one-pot, three-compo...
An unexpected rhodium-catalyzed regioselective C–H chlorination of 7-azaindoles was developed using ...
An efficient Rh(III)-catalyzed 7-azaindole synthesis was developed via C-H activation/annulative cou...
Synthetic methods used for the preparation of azaindoles are described in this article. Applications...
Tzvetkov NT, Neumann B, Stammler H-G, Antonov L. A simple approach to multifunctionalized N1-alkylat...
An efficient and practical route to 7-azaindole framework has been developed by one-pot, three-compo...
Five protocols were first compared for the copper-catalyzed C-N bond formation between 7-azaindole a...
A versatile synthesis of 7-azaindoles from substituted 2-fluoropyridines is described. C3-metalation...
By direct coupling 7-azaindole and cyclic imines, such as 3,4-dihydroisoquinoline, 6,7-dihydrothieno...
Azaindoles are rare in nature but extremely attractive for drug discovery programs. Azaindoles can b...
La séquence ihDA/rDA est une transformation d’intérêt en synthèse organique en raison de la complexi...
The reactivity of N -cyanomethyl quaternary salts of 4-, 5- and 7-azaindoles towards salicylic aldeh...
Herein we report a novel iridium(III)-catalyzed ortho-mono-alkynylation of 7-azaindoles under mild c...
A series of 3-(2-haloalkenyl)-2-pyridyl-halides undergo consecutive palladium-catalysed inter- and i...
The functionalization of arenes and heterocycles via direct C-H activation is a valuable tool in med...
An efficient and practical route to 7-azaindole framework has been developed by one-pot, three-compo...
An unexpected rhodium-catalyzed regioselective C–H chlorination of 7-azaindoles was developed using ...
An efficient Rh(III)-catalyzed 7-azaindole synthesis was developed via C-H activation/annulative cou...
Synthetic methods used for the preparation of azaindoles are described in this article. Applications...
Tzvetkov NT, Neumann B, Stammler H-G, Antonov L. A simple approach to multifunctionalized N1-alkylat...
An efficient and practical route to 7-azaindole framework has been developed by one-pot, three-compo...
Five protocols were first compared for the copper-catalyzed C-N bond formation between 7-azaindole a...
A versatile synthesis of 7-azaindoles from substituted 2-fluoropyridines is described. C3-metalation...
By direct coupling 7-azaindole and cyclic imines, such as 3,4-dihydroisoquinoline, 6,7-dihydrothieno...
Azaindoles are rare in nature but extremely attractive for drug discovery programs. Azaindoles can b...
La séquence ihDA/rDA est une transformation d’intérêt en synthèse organique en raison de la complexi...
The reactivity of N -cyanomethyl quaternary salts of 4-, 5- and 7-azaindoles towards salicylic aldeh...
Herein we report a novel iridium(III)-catalyzed ortho-mono-alkynylation of 7-azaindoles under mild c...
A series of 3-(2-haloalkenyl)-2-pyridyl-halides undergo consecutive palladium-catalysed inter- and i...
The functionalization of arenes and heterocycles via direct C-H activation is a valuable tool in med...