A chiral disulfonimide-catalyzed asymmetric synthesis of δ-amino-β-keto esters via a vinylogous Mukaiyama–Mannich reaction of the Chan diene with N-Boc imines has been developed. The desired products were obtained in good to excellent yields and enantioselectivities
Part I A large number of optically active drugs and natural products contain α- functionalised keton...
Room to swing a cat: A chiral disulfonimide has been designed as a powerful new motif for asymmetric...
An asymmetric catalytic synthesis of chiral amines using a chiral base catalysed [1,3]-proton shift ...
An organocatalytic asymmetric synthesis of δ-amino-β-ketoester derivatives has been developed. A chi...
An asymmetric Mannich reaction of silyl ketene acetals with N-Boc-amino sulfones has been developed....
A new BINOL-derived chiral disulfonimide has been developed by introducing 4-methyl-3,5-dinitropheny...
A chiral disulfonimide (DSI)-catalyzed asymmetric reduction of N-alkyl imines with Hantzsch esters a...
An efficient asymmetric biomimetic transamination of α-keto esters with quinine derivatives as chira...
route to enantioenriched α-amino esters by direct reaction of α-chloroglycine ester as a practical i...
New chiral beta-(sulfonylamino)sulfinylimidates are synthesized in high overall yield and excellent ...
An asymmetric Mannich reaction has been developed to generate chiral β-amino esters in good yields w...
The first direct catalytic asymmetric synthesis of γ-amino ketones was realized by the development o...
Highly enantioselective catalytic asymmetric reactions of rationally designed α-alkylidene β-keto im...
The first decarboxylative Mannich reaction employing β-keto acids, catalyzed by cinchonine-derived b...
It takes three to make things go right: The first direct asymmetric three‐component reaction of alde...
Part I A large number of optically active drugs and natural products contain α- functionalised keton...
Room to swing a cat: A chiral disulfonimide has been designed as a powerful new motif for asymmetric...
An asymmetric catalytic synthesis of chiral amines using a chiral base catalysed [1,3]-proton shift ...
An organocatalytic asymmetric synthesis of δ-amino-β-ketoester derivatives has been developed. A chi...
An asymmetric Mannich reaction of silyl ketene acetals with N-Boc-amino sulfones has been developed....
A new BINOL-derived chiral disulfonimide has been developed by introducing 4-methyl-3,5-dinitropheny...
A chiral disulfonimide (DSI)-catalyzed asymmetric reduction of N-alkyl imines with Hantzsch esters a...
An efficient asymmetric biomimetic transamination of α-keto esters with quinine derivatives as chira...
route to enantioenriched α-amino esters by direct reaction of α-chloroglycine ester as a practical i...
New chiral beta-(sulfonylamino)sulfinylimidates are synthesized in high overall yield and excellent ...
An asymmetric Mannich reaction has been developed to generate chiral β-amino esters in good yields w...
The first direct catalytic asymmetric synthesis of γ-amino ketones was realized by the development o...
Highly enantioselective catalytic asymmetric reactions of rationally designed α-alkylidene β-keto im...
The first decarboxylative Mannich reaction employing β-keto acids, catalyzed by cinchonine-derived b...
It takes three to make things go right: The first direct asymmetric three‐component reaction of alde...
Part I A large number of optically active drugs and natural products contain α- functionalised keton...
Room to swing a cat: A chiral disulfonimide has been designed as a powerful new motif for asymmetric...
An asymmetric catalytic synthesis of chiral amines using a chiral base catalysed [1,3]-proton shift ...