Here we report a new catalytic asymmetric synthesis of oxazolidin-2-ones 4 and Cbz-protected 1,2-amino alcohols 5. Our sequence is based on the chemistry of previously unknown 5-acyloxy-oxazolidin-2-ones, which are obtained via proline-catalyzed direct asymmetric three-component Mannich reaction and Baeyer-Villiger oxidatio
Tetrazole and acylsulfonamide organocatalysts derived from proline have been synthesised and applied...
The first organocatalytic Mannich reaction of 5H-oxazol-4-ones with various readily prepared aryl- a...
The 1,2-diamine (vicinal diamine) motif is present in a number of natural products with interesting ...
Here we report a new catalytic asymmetric synthesis of oxazolidin-2-ones 4 and Cbz-protected 1,2-ami...
We have developed proline-catalyzed direct asymmetric three-component Mannich reactions of ketones, ...
Small organic molecules recently emerged as a third class of broadly useful asymmetric catalysts tha...
This protocol describes a procedure for the synthesis of α, β-branched-b-amino aldehydes via Proline...
Mannich reaction occuring among ketone, aldehyde, and amine is one of the ways of a synthesis of bio...
A highly enantioselective catalytic route to carbamate- and benzoate-protected β-amino aldehydes and...
This account focuses on novel amine-catalyzed reactions recently discovered in our laboratories. Amo...
It is shown that racemic oxazolones are excellent reagents for the synthesis of chiral quaternary am...
A variety of (R)-phenylglycinol-derived oxazolopiperidone lactams 1-14 were converted to linear-chai...
A variety of (R)-phenylglycinol-derived oxazolopiperidone lactams 1-14 were converted to linear-chai...
Tetrazole and acylsulfonamide organocatalysts derived from proline have been synthesised and applied...
The first organocatalytic Mannich reaction of 5H-oxazol-4-ones with various readily prepared aryl- a...
Tetrazole and acylsulfonamide organocatalysts derived from proline have been synthesised and applied...
The first organocatalytic Mannich reaction of 5H-oxazol-4-ones with various readily prepared aryl- a...
The 1,2-diamine (vicinal diamine) motif is present in a number of natural products with interesting ...
Here we report a new catalytic asymmetric synthesis of oxazolidin-2-ones 4 and Cbz-protected 1,2-ami...
We have developed proline-catalyzed direct asymmetric three-component Mannich reactions of ketones, ...
Small organic molecules recently emerged as a third class of broadly useful asymmetric catalysts tha...
This protocol describes a procedure for the synthesis of α, β-branched-b-amino aldehydes via Proline...
Mannich reaction occuring among ketone, aldehyde, and amine is one of the ways of a synthesis of bio...
A highly enantioselective catalytic route to carbamate- and benzoate-protected β-amino aldehydes and...
This account focuses on novel amine-catalyzed reactions recently discovered in our laboratories. Amo...
It is shown that racemic oxazolones are excellent reagents for the synthesis of chiral quaternary am...
A variety of (R)-phenylglycinol-derived oxazolopiperidone lactams 1-14 were converted to linear-chai...
A variety of (R)-phenylglycinol-derived oxazolopiperidone lactams 1-14 were converted to linear-chai...
Tetrazole and acylsulfonamide organocatalysts derived from proline have been synthesised and applied...
The first organocatalytic Mannich reaction of 5H-oxazol-4-ones with various readily prepared aryl- a...
Tetrazole and acylsulfonamide organocatalysts derived from proline have been synthesised and applied...
The first organocatalytic Mannich reaction of 5H-oxazol-4-ones with various readily prepared aryl- a...
The 1,2-diamine (vicinal diamine) motif is present in a number of natural products with interesting ...