A rapid and simple procedure was devised for the synthesis of multifunctionalized cyclic β-amino esters and γ-amino alcohols via the 1,3-dipolar cycloaddition of nitrile oxides to β-aminocyclopentenecarboxylates. The opening of the isoxazoline reductive ring to the corresponding highly functionalized 2-aminocyclopentanecarboxylates occurred stereoselectively with good yields
Cu(I) catalyzed 3+2 cycloaddition of in situ generated N α-Fmoc/Boc/Z-protected amino alkyl nitrile...
Novel beta-aminocyclobutanecarboxylic acid derivatives were prepared via a sequential solvent-free a...
License, which permits unrestricted use, distribution, and reproduction in any medium, provided the ...
The present account illustrates the syntheses of isoxazoline- based amino acids by the cycloadditio...
Fluorinated highly functionalized cispentacin derivatives were synthetised starting from an unsatur...
AbstractA collection of isoxazoles derivatives has been efficiently synthesized in three steps. The ...
1,3-dipolar cycloaddition of arylnitrile oxides with allyl ester prepared from eugenol afforded new ...
Highly functionalized b-aminocyclohexanecarboxylate regio- and stereoisomers were synthesized from ...
Isoxazoline γ-lactams are prepared starting from the regioisomeric cycloadducts of benzonitrile oxid...
A new protocol for synthesizing different functionalized isoxazoles is provided. Carbamoylnitrile ox...
An efficient modular approach toward medicinally important 5-acylamino-4,5-isoxazolines via the 1,3-...
Abstract3,6-Dimethyl-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4(5H)-one 3 was prepared by an intramolecu...
In this paper, we report the regioselective synthesis of 3,5‐disubstituted isoxazoles by 1,3‐dipolar...
Difunctionalized cispentacin derivatives with two new stereogenic centres have been synthesized from...
Aminobenzaldehydes bearing a pendant 3,5-dinitrophenyl group react thermally with N-substituted α-am...
Cu(I) catalyzed 3+2 cycloaddition of in situ generated N α-Fmoc/Boc/Z-protected amino alkyl nitrile...
Novel beta-aminocyclobutanecarboxylic acid derivatives were prepared via a sequential solvent-free a...
License, which permits unrestricted use, distribution, and reproduction in any medium, provided the ...
The present account illustrates the syntheses of isoxazoline- based amino acids by the cycloadditio...
Fluorinated highly functionalized cispentacin derivatives were synthetised starting from an unsatur...
AbstractA collection of isoxazoles derivatives has been efficiently synthesized in three steps. The ...
1,3-dipolar cycloaddition of arylnitrile oxides with allyl ester prepared from eugenol afforded new ...
Highly functionalized b-aminocyclohexanecarboxylate regio- and stereoisomers were synthesized from ...
Isoxazoline γ-lactams are prepared starting from the regioisomeric cycloadducts of benzonitrile oxid...
A new protocol for synthesizing different functionalized isoxazoles is provided. Carbamoylnitrile ox...
An efficient modular approach toward medicinally important 5-acylamino-4,5-isoxazolines via the 1,3-...
Abstract3,6-Dimethyl-1-phenyl-1H-pyrazolo[3,4-d]pyrimidin-4(5H)-one 3 was prepared by an intramolecu...
In this paper, we report the regioselective synthesis of 3,5‐disubstituted isoxazoles by 1,3‐dipolar...
Difunctionalized cispentacin derivatives with two new stereogenic centres have been synthesized from...
Aminobenzaldehydes bearing a pendant 3,5-dinitrophenyl group react thermally with N-substituted α-am...
Cu(I) catalyzed 3+2 cycloaddition of in situ generated N α-Fmoc/Boc/Z-protected amino alkyl nitrile...
Novel beta-aminocyclobutanecarboxylic acid derivatives were prepared via a sequential solvent-free a...
License, which permits unrestricted use, distribution, and reproduction in any medium, provided the ...
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