Add to ORKGAnalogs of deamino-oxytocin and deaminc-cxypressin containing a CH 1 -N H group instead of an amide bond between positions 8 and 9 were synthesized. All tested compounds exhibit significantly lowered biological activities
ABSTRACT: The synthesis of novel oxetanyl peptides, where the amide bond is replaced by a non-hydrol...
This thesis describes the design, synthesis and pharmacological profile of a library of selective ox...
In the course of our studies of hydrophobic oxytocin (OT) analogues, we newly synthesized lipidated ...
Solid phase methodology on polyamide-kieselguhr resin was used for the synthesis of six analogs of d...
The preparation of 11 new oxytocin analogs is described. The synthesis of the protected peptides wer...
The synthesis of new OT analogues bearing the following modifications: L-ŕ-t-butylglycine [Gly(Bu')]...
The synthesis of seventeen novel conformationally constrained analogues of the neurohypophyseal pept...
Eleven oxytocin analogues substituted in position 4, 5 or 9 by tetrazole analogues of amino acids we...
Some space-constraining amino acid-containing oxytocin analogues were synthesized, of which the biol...
The nonapeptide hormone oxytocin (OT) has pivotal brain roles in social recognition and interaction ...
The 4-threonine analogues of oxytocin and of mesotocin and isotocin were prepared by solid-phase syn...
It is generally accepted that the conformation of the N-terminal part of neurohypophyseal hormones a...
This thesis describes the design, synthesis and pharmacological evaluation of non-peptide based oxyt...
A previously identified, non-peptidic oxytocin (OT) receptor agonist WAY-267,464 (1) and nine novel ...
Acute and chronic pain is often treated with opioids despite the negative side effects of constipati...
ABSTRACT: The synthesis of novel oxetanyl peptides, where the amide bond is replaced by a non-hydrol...
This thesis describes the design, synthesis and pharmacological profile of a library of selective ox...
In the course of our studies of hydrophobic oxytocin (OT) analogues, we newly synthesized lipidated ...
Solid phase methodology on polyamide-kieselguhr resin was used for the synthesis of six analogs of d...
The preparation of 11 new oxytocin analogs is described. The synthesis of the protected peptides wer...
The synthesis of new OT analogues bearing the following modifications: L-ŕ-t-butylglycine [Gly(Bu')]...
The synthesis of seventeen novel conformationally constrained analogues of the neurohypophyseal pept...
Eleven oxytocin analogues substituted in position 4, 5 or 9 by tetrazole analogues of amino acids we...
Some space-constraining amino acid-containing oxytocin analogues were synthesized, of which the biol...
The nonapeptide hormone oxytocin (OT) has pivotal brain roles in social recognition and interaction ...
The 4-threonine analogues of oxytocin and of mesotocin and isotocin were prepared by solid-phase syn...
It is generally accepted that the conformation of the N-terminal part of neurohypophyseal hormones a...
This thesis describes the design, synthesis and pharmacological evaluation of non-peptide based oxyt...
A previously identified, non-peptidic oxytocin (OT) receptor agonist WAY-267,464 (1) and nine novel ...
Acute and chronic pain is often treated with opioids despite the negative side effects of constipati...
ABSTRACT: The synthesis of novel oxetanyl peptides, where the amide bond is replaced by a non-hydrol...
This thesis describes the design, synthesis and pharmacological profile of a library of selective ox...
In the course of our studies of hydrophobic oxytocin (OT) analogues, we newly synthesized lipidated ...