A One-Pot Synthesis of Triazolodiazepines
- Hooyberghs, Geert
- Van Hove, Sofie
- Jacobs, Jeroen
- Van Meervelt, Luc
- Van der Eycken, Erik
Publication date
June 2015
DOI Publisher
Wiley-VCH ISSN
1434-193X Journal
1099-0690 Citation count (estimate)
3Abstract
A one-pot sequential A3-coupling-azidation-cyclisation approach leading to potentially biologically active diazepine analogues has been developed. The implementation of the A3-coupling reaction ensures diversity. Attention is given to this so far rarely studied structural motif of fused heterocyclic diazepines.status: publishe
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