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Design of high affinity cyclic pentapeptide ligands for Κ-opioid receptors

Przydzial, M. J.
Pogozheva, Irina D.
Ho, Jeffrey C.
Bosse, Kelly E.
Sawyer, E.
Traynor, John R.
Mosberg, Henry I.

Publication date

November 2005

DOI

10.1111/j.1399-3011.2005.00295.x

Publisher

Wiley

ISSN

1397-002X

Journal

Journal of Peptide Research

Language

English

Citation count (estimate)

11

Abstract

Peer Reviewedhttp://deepblue.lib.umich.edu/bitstream/2027.42/73319/1/j.1399-3011.2005.00295.x.pd

Extracted data

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De Marco R.
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Kluczyk A.
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Anand, Jessica P.
Porter‐barrus, Vanessa R.
Waldschmidt, Helen V.
Yeomans, Larisa
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Traynor, John R.
Mosberg, Henry I.

January 2014

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Adamska Bartłomiejczyk, Anna
Kluczyk, Alicja
Janecka, Anna
DE MARCO, ROSSELLA
GENTILUCCI, LUCA

January 2017

The study reports on a series of novel cyclopeptides based on the structure Tyr-[D-Lys-Phe-Phe-Asp]N...

Synthesis, biological evaluation, and SAR studies of 14β-phenylacetyl substituted 17-cyclopropylmethyl-7, 8-dihydronoroxymorphinones derivatives : Ligands with mixed NOP and opioid receptor profile

Kumar, Vinod
Polgar, Willma E.
Cami-Kobeci, Gerta
Thomas, Mark P.
Khroyan, Taline V.
Toll, Lawrence
Husbands, Stephen M.

September 2018

© 2018 Kumar, Polgar, Cami-Kobeci, Thomas, Khroyan, Toll and Husbands.A series of 14β-acyl substitut...

Development of a model for the δ-opioid receptor pharmacophore: 3. Comparison of the cyclic tetrapeptide Tyr-c[ D -Cys-Phe- D -Pen] OH with other conformationally constrained δ-receptor selective ligands

Lomize, Andrei L.
Pogozheva, Irina D.
Mosberg, Henry I.

February 1996

We have previously proposed a model of the δ-opioid receptor bound conformation for the cyclic tetra...

Development of functionally selective, small molecule agonists at kappa opioid receptors

Zhou, L.
Lovell, K.M.
Frankowski, K.J.
Slauson, S.R.
Phillips, A.M.
Streicher, J.M.
Stahl, E.
Schmid, C.L.
Hodde, P.
Madoux, F.
Cameron, M.D.
Prisinzano, T.E.
Aubé, J.
Bohn, L.M.

January 2013

The kappa opioid receptor (KOR) is widely expressed in the CNS and can serve as a means to modulate ...