Add to ORKGThe thermolysis of (3R,9bS)-5-oxo-2,3,5,9b-tetrahydrothiazolo[2,3-a]isoindole-3-carboxylic acids in Ac2O led to novel 3-methylene-2,5-dioxo-3H,9bH-oxazolo[2,3-a]isoindoles and chiral (9bS)-5-oxo-2,3,5,9b-tetrahydrothiazolo[2,3-a]isoindoles were obtained on FVP. Starting from -cysteine methyl ester (3R,10bR)-5-oxo-2,3-dihydro-10bH-[1.3]thiazolo[3,2-c][1,3]benzoxazines were obtained as single stereoisomers. The thermolysis of (3R,10bR)-5-oxo-2,3-dihydro-10bH-[1.3]thiazolo[3,2-c][1,3]benzoxazine-3-carboxylic acid in Ac2O gave 5-acetyl-2-phenyl-2,3-dihydrothiazole. The structures of methyl (3R,9bS)-5-oxo-2,3,5,9b-tetrahydrothiazolo[2,3-a]isoindole-3-carboxylate 1a and methyl (2R,4R)-N-chlorocarbonyl-2-(2-hydroxyphenyl)thiazolidine-4-carboxylate...
Abstract Background Thiazole is a core structural motif presents in a wide range of natural products...
In this work 3-chloro-2-chlorocarbonylbenzo[b]thiophene (1) was prepared from cinnamic acid and then...
The chemistry of isothiazoles is being intensively developed, which is evidenced by the wide range o...
Novel 3-methylene-2,5-dioxo-3H,9bH-oxazolo[2,3-a]isoindoles were prepared from the thermolysis of (3...
The thermolysis of (3R,9bS)-5-oxo-2,3,5,9b-tetrahydrothiazolo[2,3-a]isoindole-3-carboxylic acids in ...
The reaction of sodium azide with 5-substituted 3-diethylamino-4-(4-methoxyphenyl)-isothiazole 1,1 d...
3-Diethylamino-4-(4-methoxyphenyl)-isothiazole 1,1-dioxide (1) was made to react with arylalkyl-and ...
811-815A focused library of thirteen compounds, 3-((1-benzyl-1H-1,2,3-triazol-4-yl)methyl)-4-arylthi...
The title compound, C10H9NO3S, was synthesized by the reaction of benzo[d]isothiazol-3(2H)-one with ...
3-Dialkylaminoisothiazole 1,1-dioxides 1 readily undergo cycloadditions with diazoalkanes 2. The rea...
The isothiazole chemistry has been some progress from the year 1956 and since then, their chemical a...
Nitrile oxides 2 reacted with 3-diethylamino-4-(4-methoxyphenyl)-isothiazole 1,1-dioxide (1) affordi...
Sixteen new isothiazoloisoxazole 1,1-dioxides, one new isothiazolotriazole and one new isothiazolopy...
Abstract: In this work 3-chloro-2-chlorocarbonylbenzo[b]thiophene (1) was prepared from cinnamic aci...
From isothiazoles to new or known heterocycles via cycloaddition reactionsThe synthesis and chemical...
Abstract Background Thiazole is a core structural motif presents in a wide range of natural products...
In this work 3-chloro-2-chlorocarbonylbenzo[b]thiophene (1) was prepared from cinnamic acid and then...
The chemistry of isothiazoles is being intensively developed, which is evidenced by the wide range o...
Novel 3-methylene-2,5-dioxo-3H,9bH-oxazolo[2,3-a]isoindoles were prepared from the thermolysis of (3...
The thermolysis of (3R,9bS)-5-oxo-2,3,5,9b-tetrahydrothiazolo[2,3-a]isoindole-3-carboxylic acids in ...
The reaction of sodium azide with 5-substituted 3-diethylamino-4-(4-methoxyphenyl)-isothiazole 1,1 d...
3-Diethylamino-4-(4-methoxyphenyl)-isothiazole 1,1-dioxide (1) was made to react with arylalkyl-and ...
811-815A focused library of thirteen compounds, 3-((1-benzyl-1H-1,2,3-triazol-4-yl)methyl)-4-arylthi...
The title compound, C10H9NO3S, was synthesized by the reaction of benzo[d]isothiazol-3(2H)-one with ...
3-Dialkylaminoisothiazole 1,1-dioxides 1 readily undergo cycloadditions with diazoalkanes 2. The rea...
The isothiazole chemistry has been some progress from the year 1956 and since then, their chemical a...
Nitrile oxides 2 reacted with 3-diethylamino-4-(4-methoxyphenyl)-isothiazole 1,1-dioxide (1) affordi...
Sixteen new isothiazoloisoxazole 1,1-dioxides, one new isothiazolotriazole and one new isothiazolopy...
Abstract: In this work 3-chloro-2-chlorocarbonylbenzo[b]thiophene (1) was prepared from cinnamic aci...
From isothiazoles to new or known heterocycles via cycloaddition reactionsThe synthesis and chemical...
Abstract Background Thiazole is a core structural motif presents in a wide range of natural products...
In this work 3-chloro-2-chlorocarbonylbenzo[b]thiophene (1) was prepared from cinnamic acid and then...
The chemistry of isothiazoles is being intensively developed, which is evidenced by the wide range o...