Structure based design of simplified analogues of insect kinins

Kamoune, Laïla
De Borggraeve, Wim
Verbist, BMP
Vanden Broeck, Jozef
Coast, GM
Compernolle, Frans
Hoornaert, Georges

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Publication date

January 2005

DOI

10.1016/j.tet.2005.07.085

Publisher

Elsevier BV

Journal

Tetrahedron

Abstract

Based on a receptor interaction model, simplified analogues of insect kinins were prepared. The compounds were templated on a conformationally restricted amino piperidinone carboxylate scaffold. The conformation of the analogues was studied by NMR and the biological activity of the compounds was tested in a bio-assay. (c) 2005 Elsevier Ltd. All rights reserved.status: publishe

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Structure based design of simplified analogues of insect kinins

Abstract

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Structure based design of simplified analogues of insect kinins

Abstract

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