Benzotriazole-Assisted Thioacylation
- Katritzky, A.R.
- Witek, R.M.
- Rodriguez-Garcia, V.
- Mohapatra, P.P.
- Rogers, J.W.
- Cusido, J.
- Abdel-Fattah, A.A.A.
- Steel, P.J.
DOIAbstract
Benzotriazole reagents for thioacylation (RCSBt), thiocarbamoylation (RR'NCSBt), aryl/alkoxythioacylation (ROCSBt), and aryl/alkylthiothioacylation (RSCSBt) are synthesized, and their utility assessed by syntheses of representative heteroaryl thioureas 3a–g, thioamides 15a–s, thionoesters 16a– h, thiocarbamates 17a–e, dithiocarbamates 18a–d, thiocarbonates 19a–c, and dithiocarbonates 20a–c
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