Novel quinolone substituted urea and thiourea derivatives as anti-microbial and anti-cancer agents : design, synthesis and biological screening.

In vitro metabolism of tetrazole aminoquinolines and derivatives of metergoline and fusidic acid

Njoroge, Mathew

January 2014

Includes bibliographical references.Drug metabolism is recognised as a key component of the drug dis...

The SYNTHESIS, SCREENING OF NOVEL 1-SUBSTITUTED-3-(4-OXO-2-PHENYLQUINAZOLIN-3(4H)-YL) UREA AND THIOUREA ANALOGUES AS POTENT ANTIBACTERIALS

DHOKALE, SANDHYA R.
THAKAR, SNEHAL R.
BANSODE, DEEPALI A.
MAHADIK, KAKASAHEB R.

November 2019

Objective: The proposed study is an attempt to determine antibacterial activity of synthesized novel...

Derivatives of quinoxaline-2-carboxylic acid as potential antimicrobial compounds

Bouz, Sarah

January 2019

(ENGLISH) Charles University Faculty of Pharmacy in Hradec Králové Department of Pharmaceutical Chem...

Synthesis and biological evaluation of dihydropyrimidinone derivatives as a promising antimicrobial agents.

Muzenda, Wadzanai Janet.

January 2014

M. Pharm. University of KwaZulu-Natal, Durban 2014.Abstract available in PDF file

Synthesis, characterization and bioactivity of quinoxaline and benzimidazole derivatives.

Shintre, Suhas Ashok.

January 2016

Doctor of Philosophy in Chemistry. University of KwaZulu-Natal, Westville 2016.Abstract available in...

Synthesis, characterisation and biological studies of novel pyrimidine derivatives.

Aremu, Oluwole Samuel.

January 2016

Doctor of Philosophy in Chemistry. University of Kwa-Zulu Natal, Durban 2016.Abstract available in P...

Synthesis, characterisation and antibacterial activity of substituted 2-quinoline thiosemicarbazones.

Shezi, Siboniso Sibusiso.

January 2017

Masters Degree. University of KwaZulu-Natal, Durban.Fifteen quinoline-2-thiosemicarbazone hybrid der...

Synthesis and evaluation of hybrid compounds based on antimalarial and anticancer pharmacophores

Nair, Shankari

January 2012

Includes bibliographical references.Malaria stills remains one of the leading causes of death in sub...

SYNTHESIS AND BIOLOGICAL APPLICATIONS OF SOME NOVEL UREA AND THIOUREA-QUINOLINE DERIVATIVES

Jaarouf Alkaabi, Aysha Mohammed Subaih

April 2019

Extensive literature survey reveals that 8-Hydroxyquinoline (8-HQ), urea, thiourea and piperazine ex...

Synthesis and Structure-Activity Relationships of New Antibacterials against Methicillin- Resistant Staphylococcus aureus and Mycobacterium tuberculosis

Majed, Hiwa H

January 2020

Before the discovery of antibiotics, bacterial infections were a major cause of human death and suff...

Design, synthesis, and biological evaluation of novel quinoline-based molecules with potential anticancer activity

Amoozgar, Zohreh

January 2007

Quinolone derivatives have recently been introduced as inhibitors of eukaryotic topisomerase-II with...

Studies on the synthesis, cyclodextrin inclusion and biological activity of ajoene analogues as potentially novel anti-cancer agents

Qwebani, Tozama

January 2009

Includes bibliographical references (leaves 107-111).The first part of the thesis describes synthesi...

Exploring the potential of chloroquine and quinacrine derivatives as new antiprotozoal and tumour drug resistance reversal agents

Haupt, Hayley Claire

January 2002

Bibliography: leaves 108-113.Compounds containing the quinoline and acridine moieties have been util...

Molecular Design, Synthesis, Characterization & In-Vitro Biological Evaluation of Some Substituted Quinoxaline-2(1h) One Derivatives.

Parvathi Devi, R

April 2012

Medicinal Chemistry is a science whose roots lie in all branches of Chemistry and Biology. The pract...

Synthesis, characterization and evaluation of antibacterial, antidiabetic and toxicological profiles of newly-derived therapeutic agents.

Gannimani, Ramesh.

January 2016

Doctor of Philosophy in Biochemistry. University of KwaZulu-Natal, Durban 2016.Abstract available in...

In vitro metabolism of tetrazole aminoquinolines and derivatives of metergoline and fusidic acid

Njoroge, Mathew

January 2014

Includes bibliographical references.Drug metabolism is recognised as a key component of the drug dis...

The SYNTHESIS, SCREENING OF NOVEL 1-SUBSTITUTED-3-(4-OXO-2-PHENYLQUINAZOLIN-3(4H)-YL) UREA AND THIOUREA ANALOGUES AS POTENT ANTIBACTERIALS

DHOKALE, SANDHYA R.
THAKAR, SNEHAL R.
BANSODE, DEEPALI A.
MAHADIK, KAKASAHEB R.

November 2019

Objective: The proposed study is an attempt to determine antibacterial activity of synthesized novel...

Derivatives of quinoxaline-2-carboxylic acid as potential antimicrobial compounds

Bouz, Sarah

January 2019

(ENGLISH) Charles University Faculty of Pharmacy in Hradec Králové Department of Pharmaceutical Chem...

Synthesis and biological evaluation of dihydropyrimidinone derivatives as a promising antimicrobial agents.

Muzenda, Wadzanai Janet.

January 2014

M. Pharm. University of KwaZulu-Natal, Durban 2014.Abstract available in PDF file

Synthesis, characterization and bioactivity of quinoxaline and benzimidazole derivatives.

Shintre, Suhas Ashok.

January 2016

Doctor of Philosophy in Chemistry. University of KwaZulu-Natal, Westville 2016.Abstract available in...

Synthesis, characterisation and biological studies of novel pyrimidine derivatives.

Aremu, Oluwole Samuel.

January 2016

Doctor of Philosophy in Chemistry. University of Kwa-Zulu Natal, Durban 2016.Abstract available in P...

Synthesis, characterisation and antibacterial activity of substituted 2-quinoline thiosemicarbazones.

Shezi, Siboniso Sibusiso.

January 2017

Masters Degree. University of KwaZulu-Natal, Durban.Fifteen quinoline-2-thiosemicarbazone hybrid der...

Synthesis and evaluation of hybrid compounds based on antimalarial and anticancer pharmacophores

Nair, Shankari

January 2012

Includes bibliographical references.Malaria stills remains one of the leading causes of death in sub...

SYNTHESIS AND BIOLOGICAL APPLICATIONS OF SOME NOVEL UREA AND THIOUREA-QUINOLINE DERIVATIVES

Jaarouf Alkaabi, Aysha Mohammed Subaih

April 2019

Extensive literature survey reveals that 8-Hydroxyquinoline (8-HQ), urea, thiourea and piperazine ex...

Synthesis and Structure-Activity Relationships of New Antibacterials against Methicillin- Resistant Staphylococcus aureus and Mycobacterium tuberculosis

Majed, Hiwa H

January 2020

Before the discovery of antibiotics, bacterial infections were a major cause of human death and suff...

Design, synthesis, and biological evaluation of novel quinoline-based molecules with potential anticancer activity

Amoozgar, Zohreh

January 2007

Quinolone derivatives have recently been introduced as inhibitors of eukaryotic topisomerase-II with...

Studies on the synthesis, cyclodextrin inclusion and biological activity of ajoene analogues as potentially novel anti-cancer agents

Qwebani, Tozama

January 2009

Includes bibliographical references (leaves 107-111).The first part of the thesis describes synthesi...

Exploring the potential of chloroquine and quinacrine derivatives as new antiprotozoal and tumour drug resistance reversal agents

Haupt, Hayley Claire

January 2002

Bibliography: leaves 108-113.Compounds containing the quinoline and acridine moieties have been util...

Molecular Design, Synthesis, Characterization & In-Vitro Biological Evaluation of Some Substituted Quinoxaline-2(1h) One Derivatives.

Parvathi Devi, R

April 2012

Medicinal Chemistry is a science whose roots lie in all branches of Chemistry and Biology. The pract...

Synthesis, characterization and evaluation of antibacterial, antidiabetic and toxicological profiles of newly-derived therapeutic agents.

Gannimani, Ramesh.

January 2016

Doctor of Philosophy in Biochemistry. University of KwaZulu-Natal, Durban 2016.Abstract available in...

In vitro metabolism of tetrazole aminoquinolines and derivatives of metergoline and fusidic acid

Njoroge, Mathew

January 2014

Includes bibliographical references.Drug metabolism is recognised as a key component of the drug dis...

The SYNTHESIS, SCREENING OF NOVEL 1-SUBSTITUTED-3-(4-OXO-2-PHENYLQUINAZOLIN-3(4H)-YL) UREA AND THIOUREA ANALOGUES AS POTENT ANTIBACTERIALS

DHOKALE, SANDHYA R.
THAKAR, SNEHAL R.
BANSODE, DEEPALI A.
MAHADIK, KAKASAHEB R.

November 2019

Objective: The proposed study is an attempt to determine antibacterial activity of synthesized novel...

Derivatives of quinoxaline-2-carboxylic acid as potential antimicrobial compounds

Bouz, Sarah

January 2019

(ENGLISH) Charles University Faculty of Pharmacy in Hradec Králové Department of Pharmaceutical Chem...

Novel quinolone substituted urea and thiourea derivatives as anti-microbial and anti-cancer agents : design, synthesis and biological screening.

Abstract

Extracted data

Novel quinolone substituted urea and thiourea derivatives as anti-microbial and anti-cancer agents : design, synthesis and biological screening.

Abstract

Extracted data

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