2,3-Dihydro-1,5-benzothiazepines have been obtained through a domino process involving a Michael addition of 2-aminothiophenols to chalcones, followed by in situ cyclization. Up to 98% chemical yields have been obtained at room temperature under essentially neutral conditions by using hexafluoro-2-propanol as an efficient medium
2,3-dihydro[1,5] benzothiazepines and diazepines can be prepared by condensation of o-aminothiopheno...
The title compounds 3a-j, substituted 1,5-benzothiazepines were synthesized by the condensation of ...
The production of effective drugs has continuously been a challenging process for researchers due t...
We have developed a domino process involving the Michael addition of 2-aminothiophenols to chalcones...
A one-pot enantioselective route to N-unprotected 2,3-dihydro-1,5-benzothiazepinones, by an organoca...
The synthesis of a library of bicyclic sultams incorporating the 1,5,2-dithiazepine 1,1-dioxide moie...
A novel one-pot sulfonylation/intramolecular thia-Michael protocol is reported for the synthesis of ...
AbstractAn efficient synthesis of new derivatives of 1,5-benzothiazepine has been developed by the r...
1,5-Benzothiazepines derivatives were obtained first by starting from 1,3-diphenylpropenone derivat...
199-201<span style="font-size:14.0pt;line-height: 115%;font-family:" times="" new="" roman";mso-far...
A general procedure for the synthesis of 2-substituted tetrahydro-1,3-thiazepines by MW-assisted cyc...
A simple, convenient, and environmentally benign synthesis of 1,5-benzodiazepines is developed by c...
1,5-Benzothiazepine frameworks are highly relevant in medicinal chemistry. Reported catalytic asymme...
AbstractMichael addition reaction of 1,3-diphenyl-propenone 1a, e, and f with o-amino thiophenol in ...
A simple and elegant method for the synthesis of 1,5-benzothiazepines has been developed using di-ca...
2,3-dihydro[1,5] benzothiazepines and diazepines can be prepared by condensation of o-aminothiopheno...
The title compounds 3a-j, substituted 1,5-benzothiazepines were synthesized by the condensation of ...
The production of effective drugs has continuously been a challenging process for researchers due t...
We have developed a domino process involving the Michael addition of 2-aminothiophenols to chalcones...
A one-pot enantioselective route to N-unprotected 2,3-dihydro-1,5-benzothiazepinones, by an organoca...
The synthesis of a library of bicyclic sultams incorporating the 1,5,2-dithiazepine 1,1-dioxide moie...
A novel one-pot sulfonylation/intramolecular thia-Michael protocol is reported for the synthesis of ...
AbstractAn efficient synthesis of new derivatives of 1,5-benzothiazepine has been developed by the r...
1,5-Benzothiazepines derivatives were obtained first by starting from 1,3-diphenylpropenone derivat...
199-201<span style="font-size:14.0pt;line-height: 115%;font-family:" times="" new="" roman";mso-far...
A general procedure for the synthesis of 2-substituted tetrahydro-1,3-thiazepines by MW-assisted cyc...
A simple, convenient, and environmentally benign synthesis of 1,5-benzodiazepines is developed by c...
1,5-Benzothiazepine frameworks are highly relevant in medicinal chemistry. Reported catalytic asymme...
AbstractMichael addition reaction of 1,3-diphenyl-propenone 1a, e, and f with o-amino thiophenol in ...
A simple and elegant method for the synthesis of 1,5-benzothiazepines has been developed using di-ca...
2,3-dihydro[1,5] benzothiazepines and diazepines can be prepared by condensation of o-aminothiopheno...
The title compounds 3a-j, substituted 1,5-benzothiazepines were synthesized by the condensation of ...
The production of effective drugs has continuously been a challenging process for researchers due t...
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