Starting from isatoic anhydride and propargyl alcohols, we developed a synthetic approach to the title compounds, where the key step is an intramolecular cycloaddition of the azido group onto the acetylenic bond
Intramolecular azide cycloadditions onto the cyano group are described as a synthetic tool for a num...
A series of [1.2.4]triazolo[1,5-a][1,4]benzodiazepin-6-ones of potential pharmacological interest ha...
A novel three-step approach leading to [1,2,3]-triazolo[1,5-a][1,4] benzodiazepines in moderate to g...
A facile synthesis of [1,2,3]triazolo[1,5-a][1,4]benzodiazepines starting from isatoic anhydrides an...
A general synthetic route to the title heterocyclic compounds has been developed based on the title ...
Intramolecular 1,3-dipolar cycloaddition between an alkyne and an azide leads to a series of 1,2,3-t...
Synthesis of a series of [1,2,3] triazolo [5,1-c] [1,4]benzoxazepine derivatives have been accomplis...
Intermolecular dipolar cycloadditions between 2-methoxycarbonyl-3-thenylazide (3) and monosubstitute...
A number of 8-substituted 5-methyl[1,2,3]triazolo[1,5-a][1,4] benzodiazepin-6(4H)-ones (6) were synt...
The sequential Sonogashira coupling/intramolecular azide cyclo- addition (Huisgen cycloaddition) pro...
Starting from 2-carboxy-3-thenylazide 1 and enantiopure amines 2 as the chiral building blocks, we d...
3-Aryl substituted benzo[1,2,5]triazepin-4-ones and their pyrido counterparts have been synthesized ...
3-Aryl substituted benzo[1,2,5]triazepin-4-ones and their pyrido counterparts have been synthesized ...
3-Aryl substituted benzo[1,2,5]triazepin-4-ones and their pyrido counterparts have been synthesized ...
We review in this article some of our work which has been published over the last fifteen years in t...
Intramolecular azide cycloadditions onto the cyano group are described as a synthetic tool for a num...
A series of [1.2.4]triazolo[1,5-a][1,4]benzodiazepin-6-ones of potential pharmacological interest ha...
A novel three-step approach leading to [1,2,3]-triazolo[1,5-a][1,4] benzodiazepines in moderate to g...
A facile synthesis of [1,2,3]triazolo[1,5-a][1,4]benzodiazepines starting from isatoic anhydrides an...
A general synthetic route to the title heterocyclic compounds has been developed based on the title ...
Intramolecular 1,3-dipolar cycloaddition between an alkyne and an azide leads to a series of 1,2,3-t...
Synthesis of a series of [1,2,3] triazolo [5,1-c] [1,4]benzoxazepine derivatives have been accomplis...
Intermolecular dipolar cycloadditions between 2-methoxycarbonyl-3-thenylazide (3) and monosubstitute...
A number of 8-substituted 5-methyl[1,2,3]triazolo[1,5-a][1,4] benzodiazepin-6(4H)-ones (6) were synt...
The sequential Sonogashira coupling/intramolecular azide cyclo- addition (Huisgen cycloaddition) pro...
Starting from 2-carboxy-3-thenylazide 1 and enantiopure amines 2 as the chiral building blocks, we d...
3-Aryl substituted benzo[1,2,5]triazepin-4-ones and their pyrido counterparts have been synthesized ...
3-Aryl substituted benzo[1,2,5]triazepin-4-ones and their pyrido counterparts have been synthesized ...
3-Aryl substituted benzo[1,2,5]triazepin-4-ones and their pyrido counterparts have been synthesized ...
We review in this article some of our work which has been published over the last fifteen years in t...
Intramolecular azide cycloadditions onto the cyano group are described as a synthetic tool for a num...
A series of [1.2.4]triazolo[1,5-a][1,4]benzodiazepin-6-ones of potential pharmacological interest ha...
A novel three-step approach leading to [1,2,3]-triazolo[1,5-a][1,4] benzodiazepines in moderate to g...