Specificity of various purine inhibitors for different glycosylase-substrate combinations as determined by IC50 value.

Comparison of the amino acid compositions of GpA72 and α-Cysteine protease inhibitor.

Bina Joe (591407)
Anitha Nagaraju (641663)
Lalitha R. Gowda (641664)
Venkatesha Basrur (236779)
Belur R. Lokesh (641665)

October 2014

Comparison of the amino acid compositions of GpA72 and α-Cysteine protease inhibitor.</p

Inhibition studies of EhOASS.

Isha Nagpal (183347)
Isha Raj (183350)
Naidu Subbarao (183352)
Samudrala Gourinath (31302)

February 2012

The concentration of the inhibitor was kept at 100 µM and the readings were taken under two subst...

Design of glycosyltransferase inhibitors : serine analogues as pyrophosphate surrogates ?

Wang, Shuai
Cuesta-Seijo, José A.
Striebeck, Alexander
Lafont, Dominique
Palcic, Monica M.
Vidal, Sébastien

July 2015

International audienceMimicking the diphosphate moiety of nucleotide diphosphate sugars with serine ...

Inhibitors and probes targeting endo-glycosidases

Boer, C. de

February 2021

The chemical synthesis of inhibitors and probes targeting endo-glycosidases. </p

Direct comparison of the C1 inhibitor potentiation by test compounds with differing glycan structure.

Ann-Kathrin Schoenfeld (3269883)
Eric Lahrsen (3269880)
Susanne Alban (2339212)

October 2016

Direct comparison of the C1 inhibitor potentiation by test compounds with differing glycan struct...

Compositions of different inhibitors in corncob hydrolysate with total sugar concentration 150 g/L.

Xiang Zou (706903)
Yongkang Wang (706904)
Guangwei Tu (706905)
Zhanquan Zan (706906)
Xiaoyan Wu (235931)

March 2015

Compositions of different inhibitors in corncob hydrolysate with total sugar concentration 150 g/...

Enzyme inhibition IC50s for thrombin and other serine proteases.

Mohanram Sivaraja (2004994)
Nicola Pozzi (2866730)
Matthew Rienzo (1997911)
Kenneth Lin (1547371)
Timothy P. Shiau (2516746)
Daniel M. Clemens (5587070)
Lev Igoudin (5587073)
Piotr Zalicki (5587076)
Stephanie S. Chang (5466101)
M. Angels Estiarte (2354884)
Kevin M. Short (5587079)
David C. Williams (2680522)
Anirban Datta (225408)
Enrico Di Cera (2495530)
David B. Kita (5587082)

August 2018

Enzyme inhibition IC50s for thrombin and other serine proteases.</p

Specificity of the kinase inhibitors for CLK1, CLK2, SRPK1, SRPK2, and SRPK3.

Shinsuke Araki (491598)
Ryo Dairiki (683049)
Yusuke Nakayama (683050)
Aiko Murai (683051)
Risa Miyashita (683052)
Misa Iwatani (683053)
Toshiyuki Nomura (683054)
Osamu Nakanishi (683055)

January 2015

CLK1, SRPK1, SRPK2, and SRPK3 assays were performed with 5 µM ATP, and the CLK2 assay was perform...

vitro p-glycoprotein inhibition assays for assessment of clinical drug interaction potential of new drug candidates: a recommendation for probe substrates. Drug Metab Dispos. 2006;34(5):786–792. submit your manuscript | www.dovepress.com Dovepress Dovepre

Jarkko Rautio
Joan E. Humphreys
Lindsey O. Webster
John P. Keogh
Jeevan R. Kunta
Cosette J. Serabjit-singh
Joseph W. Polli

October 2016

Because modulation of P-glycoprotein (Pgp) through inhibition or induction can lead to drug-drug int...

Inhibitors of helicase available until now and their binding specificities.

Kaneez Fatima (625825)
Shilu Mathew (625826)
Mohd Suhail (528221)
Ashraf Ali (625827)
Ghazi Damanhouri (519678)
Esam Azhar (519677)
Ishtiaq Qadri (625828)

September 2014

Inhibitors of helicase available until now and their binding specificities.</p

Estimation of optimal substrate concentration for Mur synthetases.

Tulika Munshi (392669)
Antima Gupta (392670)
Dimitrios Evangelopoulos (392671)
Juan David Guzman (392672)
Simon Gibbons (391868)
Nicholas H. Keep (392673)
Sanjib Bhakta (106475)

March 2013

Inhibition curves obtained for MurC, MurD and MurF synthetases with (A) ATP and (B) their respect...

IC50 concentrations and maximal inhibition for WU-1 and WU-2 for class I GLUT overexpressing cells.

Monique R. Heitmeier (6686069)
Richard C. Hresko (343537)
Rachel L. Edwards (1621342)
Michael J. Prinsen (5730863)
Ma Xenia G. Ilagan (6686072)
Audrey R. Odom John (5778773)
Paul W. Hruz (343538)

May 2019

IC50 concentrations and maximal inhibition for WU-1 and WU-2 for class I GLUT overexpressing cells.<...

Studies on the Differential Specificity of Protein Kinases and Its Applications

Loog, Mart

January 2001

Protein kinases are enzymes that catalyse the phosphoryl transfer from the g-phosphate of ATP to acc...

Concentration of the inhibitors required to reduce the enzyme activity by 50%.

Mohammad Faheem (380758)
Md Tabish Rehman (380759)
Mohd Danishuddin (110825)
Asad U. Khan (110840)

February 2013

Concentration of the inhibitors required to reduce the enzyme activity by 50%.</p

Specificity of the inhibition of NEIL1.

Aaron C. Jacobs (494938)
Marcus J. Calkins (494939)
Ajit Jadhav (85100)
Dorjbal Dorjsuren (126214)
David Maloney (494940)
Anton Simeonov (85099)
Pawel Jaruga (9759)
Miral Dizdaroglu (9761)
Amanda K. McCullough (494941)
R. Stephen Lloyd (110287)

December 2013

A) Inhibition of the lyase activity of various bifunctional glycosylases with purine analogs. B) ...

Comparison of the amino acid compositions of GpA72 and α-Cysteine protease inhibitor.

Bina Joe (591407)
Anitha Nagaraju (641663)
Lalitha R. Gowda (641664)
Venkatesha Basrur (236779)
Belur R. Lokesh (641665)

October 2014

Comparison of the amino acid compositions of GpA72 and α-Cysteine protease inhibitor.</p

Inhibition studies of EhOASS.

Isha Nagpal (183347)
Isha Raj (183350)
Naidu Subbarao (183352)
Samudrala Gourinath (31302)

February 2012

The concentration of the inhibitor was kept at 100 µM and the readings were taken under two subst...

Design of glycosyltransferase inhibitors : serine analogues as pyrophosphate surrogates ?

Wang, Shuai
Cuesta-Seijo, José A.
Striebeck, Alexander
Lafont, Dominique
Palcic, Monica M.
Vidal, Sébastien

July 2015

International audienceMimicking the diphosphate moiety of nucleotide diphosphate sugars with serine ...

Inhibitors and probes targeting endo-glycosidases

Boer, C. de

February 2021

The chemical synthesis of inhibitors and probes targeting endo-glycosidases. </p

Direct comparison of the C1 inhibitor potentiation by test compounds with differing glycan structure.

Ann-Kathrin Schoenfeld (3269883)
Eric Lahrsen (3269880)
Susanne Alban (2339212)

October 2016

Direct comparison of the C1 inhibitor potentiation by test compounds with differing glycan struct...

Compositions of different inhibitors in corncob hydrolysate with total sugar concentration 150 g/L.

Xiang Zou (706903)
Yongkang Wang (706904)
Guangwei Tu (706905)
Zhanquan Zan (706906)
Xiaoyan Wu (235931)

March 2015

Compositions of different inhibitors in corncob hydrolysate with total sugar concentration 150 g/...

Enzyme inhibition IC50s for thrombin and other serine proteases.

Mohanram Sivaraja (2004994)
Nicola Pozzi (2866730)
Matthew Rienzo (1997911)
Kenneth Lin (1547371)
Timothy P. Shiau (2516746)
Daniel M. Clemens (5587070)
Lev Igoudin (5587073)
Piotr Zalicki (5587076)
Stephanie S. Chang (5466101)
M. Angels Estiarte (2354884)
Kevin M. Short (5587079)
David C. Williams (2680522)
Anirban Datta (225408)
Enrico Di Cera (2495530)
David B. Kita (5587082)

August 2018

Enzyme inhibition IC50s for thrombin and other serine proteases.</p

Specificity of the kinase inhibitors for CLK1, CLK2, SRPK1, SRPK2, and SRPK3.

Shinsuke Araki (491598)
Ryo Dairiki (683049)
Yusuke Nakayama (683050)
Aiko Murai (683051)
Risa Miyashita (683052)
Misa Iwatani (683053)
Toshiyuki Nomura (683054)
Osamu Nakanishi (683055)

January 2015

CLK1, SRPK1, SRPK2, and SRPK3 assays were performed with 5 µM ATP, and the CLK2 assay was perform...

vitro p-glycoprotein inhibition assays for assessment of clinical drug interaction potential of new drug candidates: a recommendation for probe substrates. Drug Metab Dispos. 2006;34(5):786–792. submit your manuscript | www.dovepress.com Dovepress Dovepre

Jarkko Rautio
Joan E. Humphreys
Lindsey O. Webster
John P. Keogh
Jeevan R. Kunta
Cosette J. Serabjit-singh
Joseph W. Polli

October 2016

Because modulation of P-glycoprotein (Pgp) through inhibition or induction can lead to drug-drug int...

Inhibitors of helicase available until now and their binding specificities.

Kaneez Fatima (625825)
Shilu Mathew (625826)
Mohd Suhail (528221)
Ashraf Ali (625827)
Ghazi Damanhouri (519678)
Esam Azhar (519677)
Ishtiaq Qadri (625828)

September 2014

Inhibitors of helicase available until now and their binding specificities.</p

Estimation of optimal substrate concentration for Mur synthetases.

Tulika Munshi (392669)
Antima Gupta (392670)
Dimitrios Evangelopoulos (392671)
Juan David Guzman (392672)
Simon Gibbons (391868)
Nicholas H. Keep (392673)
Sanjib Bhakta (106475)

March 2013

Inhibition curves obtained for MurC, MurD and MurF synthetases with (A) ATP and (B) their respect...

IC50 concentrations and maximal inhibition for WU-1 and WU-2 for class I GLUT overexpressing cells.

Monique R. Heitmeier (6686069)
Richard C. Hresko (343537)
Rachel L. Edwards (1621342)
Michael J. Prinsen (5730863)
Ma Xenia G. Ilagan (6686072)
Audrey R. Odom John (5778773)
Paul W. Hruz (343538)

May 2019

IC50 concentrations and maximal inhibition for WU-1 and WU-2 for class I GLUT overexpressing cells.<...

Studies on the Differential Specificity of Protein Kinases and Its Applications

Loog, Mart

January 2001

Protein kinases are enzymes that catalyse the phosphoryl transfer from the g-phosphate of ATP to acc...

Concentration of the inhibitors required to reduce the enzyme activity by 50%.

Mohammad Faheem (380758)
Md Tabish Rehman (380759)
Mohd Danishuddin (110825)
Asad U. Khan (110840)

February 2013

Concentration of the inhibitors required to reduce the enzyme activity by 50%.</p

Specificity of the inhibition of NEIL1.

Aaron C. Jacobs (494938)
Marcus J. Calkins (494939)
Ajit Jadhav (85100)
Dorjbal Dorjsuren (126214)
David Maloney (494940)
Anton Simeonov (85099)
Pawel Jaruga (9759)
Miral Dizdaroglu (9761)
Amanda K. McCullough (494941)
R. Stephen Lloyd (110287)

December 2013

A) Inhibition of the lyase activity of various bifunctional glycosylases with purine analogs. B) ...

Comparison of the amino acid compositions of GpA72 and α-Cysteine protease inhibitor.

Bina Joe (591407)
Anitha Nagaraju (641663)
Lalitha R. Gowda (641664)
Venkatesha Basrur (236779)
Belur R. Lokesh (641665)

October 2014

Comparison of the amino acid compositions of GpA72 and α-Cysteine protease inhibitor.</p

Inhibition studies of EhOASS.

Isha Nagpal (183347)
Isha Raj (183350)
Naidu Subbarao (183352)
Samudrala Gourinath (31302)

February 2012

The concentration of the inhibitor was kept at 100 µM and the readings were taken under two subst...

Design of glycosyltransferase inhibitors : serine analogues as pyrophosphate surrogates ?

Wang, Shuai
Cuesta-Seijo, José A.
Striebeck, Alexander
Lafont, Dominique
Palcic, Monica M.
Vidal, Sébastien

July 2015

International audienceMimicking the diphosphate moiety of nucleotide diphosphate sugars with serine ...

Specificity of various purine inhibitors for different glycosylase-substrate combinations as determined by IC<sub>50</sub> value.

Abstract

Extracted data

Specificity of various purine inhibitors for different glycosylase-substrate combinations as determined by IC<sub>50</sub> value.

Abstract

Extracted data

Related items

Related items