Step-economic and scalable syntheses of novel thia-azaspiro[3.4]octanes are reported. These spirocycles and some related intermediates can serve as uncharted multifunctional modules for drug discovery chemistry
MicroreviewInternational audienceThe 1-oxa-7-azaspiro[5.5]undecane, 1-oxa-6-azaspiro[4.5]decane, 1-o...
The first objective of this work was to synthesize certain substituted cyclohexanespiropiperidines (...
Graduation date: 2013Azaspiracid-1, a novel marine toxin that contains 9 rings and 20 stereogenic ce...
New classes of thia/oxa-azaspiro[3.4]octanes are synthesized through the implementation of robust an...
The preparation of versatile azaspiro[3.3]heptanes carrying multiple exit vectors is disclosed. Expe...
Multicomponent condensation of N-diphenylphosphinoylimines, alkynes, zirconocene hydrochloride, and ...
Recently we have developed a methodology for the synthesis of spirocyclohexadienones1,2,3. These com...
Azaspirocycles are found as structural motif in a number of highly interesting natural products. In ...
International audienceFrom their discovery in the late 1960s, iminosugars have undergone an expansio...
Present communication deals with the synthesis and characterization of various spiro thiazolinone he...
A detailed synthesis of spirocyclic amine analogs is described for the first tim
Synthetic approaches toward multigram preparation of spirocyclic α,α-disubstituted pyrrolidines from...
A solution-phase parallel synthesis of pharmaceutically important azaspiro[4.5]trienones has been d...
A convergent and stereoselective synthesis of 1-oxa-7-azaspiro[5.5]undecane is described. This funct...
A facile, efficient and unprecedented method for the synthesis of spiro-2H-pyrroles is reported. Whe...
MicroreviewInternational audienceThe 1-oxa-7-azaspiro[5.5]undecane, 1-oxa-6-azaspiro[4.5]decane, 1-o...
The first objective of this work was to synthesize certain substituted cyclohexanespiropiperidines (...
Graduation date: 2013Azaspiracid-1, a novel marine toxin that contains 9 rings and 20 stereogenic ce...
New classes of thia/oxa-azaspiro[3.4]octanes are synthesized through the implementation of robust an...
The preparation of versatile azaspiro[3.3]heptanes carrying multiple exit vectors is disclosed. Expe...
Multicomponent condensation of N-diphenylphosphinoylimines, alkynes, zirconocene hydrochloride, and ...
Recently we have developed a methodology for the synthesis of spirocyclohexadienones1,2,3. These com...
Azaspirocycles are found as structural motif in a number of highly interesting natural products. In ...
International audienceFrom their discovery in the late 1960s, iminosugars have undergone an expansio...
Present communication deals with the synthesis and characterization of various spiro thiazolinone he...
A detailed synthesis of spirocyclic amine analogs is described for the first tim
Synthetic approaches toward multigram preparation of spirocyclic α,α-disubstituted pyrrolidines from...
A solution-phase parallel synthesis of pharmaceutically important azaspiro[4.5]trienones has been d...
A convergent and stereoselective synthesis of 1-oxa-7-azaspiro[5.5]undecane is described. This funct...
A facile, efficient and unprecedented method for the synthesis of spiro-2H-pyrroles is reported. Whe...
MicroreviewInternational audienceThe 1-oxa-7-azaspiro[5.5]undecane, 1-oxa-6-azaspiro[4.5]decane, 1-o...
The first objective of this work was to synthesize certain substituted cyclohexanespiropiperidines (...
Graduation date: 2013Azaspiracid-1, a novel marine toxin that contains 9 rings and 20 stereogenic ce...
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