<p>Inhibitory activity (IC<sub>50</sub>, μM) against MAO-A and -B and selectivity index for LSD1.</p
<p>*- the K<sub>i</sub> values were calculated using the online IC<sub>50</sub>-to-<i>K<sub>i</sub><...
<p>Molecular descriptors highly correlated with OCT1 activity inhibition for BIMs (r>0.90).</p
<p>The IC<sub>50</sub> stands for the compound concentration where half-maximal inhibition is observ...
<p>Inhibition potencies of 1,2-diarylethylamines as monoamine transporter reuptake inhibitors.</p
<p>The number of compounds found to demonstrate inhibition at 10μM overall and with respect to the t...
<p>All IC<sub>50</sub> values shown are the means ± SEM from five experiments.</p>a<p>Percentage inh...
Inhibitory activity of selected hits against MG1655 in the presence and absence of 4-NQO.</p
<div><p>Post-translational modifications of histone play important roles in gene transcription. Aber...
Post-translational modifications of histone play important roles in gene transcription. Aberrant met...
© 2020 Elsevier LtdThe inhibitory activity of monoamine oxidase A (MAO-A) was investigated as 4D- Qu...
The pure four diastereomers (11a-d) of trans-benzyl (1-((4-(2-aminocyclopropyl)phenyl)amino)-1-oxo-3...
The actions of many drugs involve enzyme inhibition. This is exemplified by the inhibitors of monoam...
The actions of many drugs involve enzyme inhibition. This is exemplified by the inhibitors of monoam...
The pure four diastereomers (11a-d) of trans-benzyl (1-((4-(2-aminocyclopropyl)phenyl)amino)-1-oxo-3...
<p>A) CGP-74514A, B) P2, C) P6, D) P7, E) P8 compared to no inhibitor (gray squares) or no enzyme (g...
<p>*- the K<sub>i</sub> values were calculated using the online IC<sub>50</sub>-to-<i>K<sub>i</sub><...
<p>Molecular descriptors highly correlated with OCT1 activity inhibition for BIMs (r>0.90).</p
<p>The IC<sub>50</sub> stands for the compound concentration where half-maximal inhibition is observ...
<p>Inhibition potencies of 1,2-diarylethylamines as monoamine transporter reuptake inhibitors.</p
<p>The number of compounds found to demonstrate inhibition at 10μM overall and with respect to the t...
<p>All IC<sub>50</sub> values shown are the means ± SEM from five experiments.</p>a<p>Percentage inh...
Inhibitory activity of selected hits against MG1655 in the presence and absence of 4-NQO.</p
<div><p>Post-translational modifications of histone play important roles in gene transcription. Aber...
Post-translational modifications of histone play important roles in gene transcription. Aberrant met...
© 2020 Elsevier LtdThe inhibitory activity of monoamine oxidase A (MAO-A) was investigated as 4D- Qu...
The pure four diastereomers (11a-d) of trans-benzyl (1-((4-(2-aminocyclopropyl)phenyl)amino)-1-oxo-3...
The actions of many drugs involve enzyme inhibition. This is exemplified by the inhibitors of monoam...
The actions of many drugs involve enzyme inhibition. This is exemplified by the inhibitors of monoam...
The pure four diastereomers (11a-d) of trans-benzyl (1-((4-(2-aminocyclopropyl)phenyl)amino)-1-oxo-3...
<p>A) CGP-74514A, B) P2, C) P6, D) P7, E) P8 compared to no inhibitor (gray squares) or no enzyme (g...
<p>*- the K<sub>i</sub> values were calculated using the online IC<sub>50</sub>-to-<i>K<sub>i</sub><...
<p>Molecular descriptors highly correlated with OCT1 activity inhibition for BIMs (r>0.90).</p
<p>The IC<sub>50</sub> stands for the compound concentration where half-maximal inhibition is observ...
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