A solution phase combinatorial synthesis of aryl piperazines 1 and 2 is described based on the S(N)Ar reaction and Schotten-Baumann acylation. The use of excess reagent is allowed and pure arylpiperazines 1 and 2 were obtained by simple acid/base washing
A simple and straightforward methodology for the parallel, solution-phase synthesis of novel 4-dialk...
The need to find more efficient and cost-effective methods of drug development has led pharmaceutica...
Peptides containing N2-acyl piperazic or 1,6-dehydropiperazic acids can be formed efficiently via a...
Abstract: The palladium-catalyzed coupling of amines and aryl halides or aryl alcohol derivatives ha...
The first application of aziridine aldehyde dimers in solid-phase synthesis is reported. The solid-s...
Structurally diverse amino acids were prepared as versatile synthons for combinatorial chemistry. Us...
A cascade, metal promoted transformations utilizing chloro allenylamide, primary amine and aryl iodi...
[[abstract]]A series of monosubstituted piperazine derivatives were obtained by the reaction of pipe...
A simple and efficient one-step procedure is described for the synthesis of a number of symmetrical ...
[[abstract]]A series of monosubstituted piperazine derivatives were obtained by the reaction of pipe...
Piperazines are widely used as central elements in the construction of bioactive molecules. Herein, ...
An efficient one-pot synthesis is described for the preparation of 1,4-disubstituted piperazine-2,5-...
A synthetic methodology to prepare collections of trisubstituted aryl 1,3,5-triazines with broad str...
A simple and straightforward methodology for the parallel, solution-phase synthesis of novel 4-dialk...
An efficient solution-phase synthesis of aza-diketopiperazines (aza-DKP, triazinediones) is reported...
A simple and straightforward methodology for the parallel, solution-phase synthesis of novel 4-dialk...
The need to find more efficient and cost-effective methods of drug development has led pharmaceutica...
Peptides containing N2-acyl piperazic or 1,6-dehydropiperazic acids can be formed efficiently via a...
Abstract: The palladium-catalyzed coupling of amines and aryl halides or aryl alcohol derivatives ha...
The first application of aziridine aldehyde dimers in solid-phase synthesis is reported. The solid-s...
Structurally diverse amino acids were prepared as versatile synthons for combinatorial chemistry. Us...
A cascade, metal promoted transformations utilizing chloro allenylamide, primary amine and aryl iodi...
[[abstract]]A series of monosubstituted piperazine derivatives were obtained by the reaction of pipe...
A simple and efficient one-step procedure is described for the synthesis of a number of symmetrical ...
[[abstract]]A series of monosubstituted piperazine derivatives were obtained by the reaction of pipe...
Piperazines are widely used as central elements in the construction of bioactive molecules. Herein, ...
An efficient one-pot synthesis is described for the preparation of 1,4-disubstituted piperazine-2,5-...
A synthetic methodology to prepare collections of trisubstituted aryl 1,3,5-triazines with broad str...
A simple and straightforward methodology for the parallel, solution-phase synthesis of novel 4-dialk...
An efficient solution-phase synthesis of aza-diketopiperazines (aza-DKP, triazinediones) is reported...
A simple and straightforward methodology for the parallel, solution-phase synthesis of novel 4-dialk...
The need to find more efficient and cost-effective methods of drug development has led pharmaceutica...
Peptides containing N2-acyl piperazic or 1,6-dehydropiperazic acids can be formed efficiently via a...
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