The invention relates to a method of preparing a reaction product such as a primary amide, by means of two reagents A and B, which reagents form a salt that impedes fast conversion. The concentrations of the reagent A and the reagent B are chosen such that they comply with formula (I) wherein [A]T represents the concentration of the first reagent A in relation to the total volume taken up by the reagents A, B, and the solvent.Applied Science
Amide linkages are present in key natural products and in many biologically active molecules. Theref...
The present invention relates to a process for the amidation of C-terminal esters or acids of peptid...
This work focuses on the Lipase-catalyzed synthesis of esters and amides of great interest for the c...
The invention relates to a method of preparing a reaction product such as a primary amide, by means ...
Abstract The synthesis of the amide bond between an amine and a carboxylic acid is one of the most s...
N-Alkyl carbamates of primary amines are easily converted into amides under treatment with Grignard ...
A lipase-catalyzed procedure is described for the one-pot conversion of carboxylic acids into substi...
Despite the amide formation reaction being a key reaction in organic chemistry, the direct amide for...
Amide bond is a special structure that can exhibit high physiological activity. The most ideal way t...
An efficient method has been developed for the preparation of yet unknown acyclic mixed anhydrides o...
Current methods for constructing amide bonds join amines and carboxylic acids by dehydrative couplin...
Amides are important organic compounds that are widely applied in medicine, biochemistry, and materi...
A symmetric diketopiperazine scaffold 2 has been prepared in a very simple two-step procedure from 1...
B(OCH<sub>2</sub>CF<sub>3</sub>)<sub>3</sub>, prepared from readily available B<sub>2</sub>O<sub>3<...
A general method for the synthesis of amides involving the direct coupling of alkali metal carboxyla...
Amide linkages are present in key natural products and in many biologically active molecules. Theref...
The present invention relates to a process for the amidation of C-terminal esters or acids of peptid...
This work focuses on the Lipase-catalyzed synthesis of esters and amides of great interest for the c...
The invention relates to a method of preparing a reaction product such as a primary amide, by means ...
Abstract The synthesis of the amide bond between an amine and a carboxylic acid is one of the most s...
N-Alkyl carbamates of primary amines are easily converted into amides under treatment with Grignard ...
A lipase-catalyzed procedure is described for the one-pot conversion of carboxylic acids into substi...
Despite the amide formation reaction being a key reaction in organic chemistry, the direct amide for...
Amide bond is a special structure that can exhibit high physiological activity. The most ideal way t...
An efficient method has been developed for the preparation of yet unknown acyclic mixed anhydrides o...
Current methods for constructing amide bonds join amines and carboxylic acids by dehydrative couplin...
Amides are important organic compounds that are widely applied in medicine, biochemistry, and materi...
A symmetric diketopiperazine scaffold 2 has been prepared in a very simple two-step procedure from 1...
B(OCH<sub>2</sub>CF<sub>3</sub>)<sub>3</sub>, prepared from readily available B<sub>2</sub>O<sub>3<...
A general method for the synthesis of amides involving the direct coupling of alkali metal carboxyla...
Amide linkages are present in key natural products and in many biologically active molecules. Theref...
The present invention relates to a process for the amidation of C-terminal esters or acids of peptid...
This work focuses on the Lipase-catalyzed synthesis of esters and amides of great interest for the c...